SCHEMBL8035683

SCHEMBL8035683

COCCCN(C(=O)NC1CC1)C(=O)c1c(C(F)(F)F)cc(O)c(O)c1[N+](=O)[O-]

nearest known ligand 0.32

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SMYD3 Q9H7B4 1/20 0.32
TAS1R3 Q7RTX0 1/20 0.32
TAS1R1 Q7RTX1 1/20 0.32
TAS1R2 Q8TE23 1/20 0.32
SLC6A2 P23975 2/20 0.32
SLC6A4 P31645 2/20 0.32
USP30 Q70CQ3 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C19 P33261 1/20 0.31
DCUN1D1 Q96GG9 1/20 0.31
COMT P21964 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8040084 0.91 ALDH1A1 (0.33) TAS1R3TAS1R1TAS1R2SLC6A2SLC6A4
SCHEMBL8041249 0.81 TAS1R3 (0.35) TAS1R3TAS1R1TAS1R2COMT
SCHEMBL8025508 0.77 ALDH1A1 (0.37) COMT
SCHEMBL8037861 0.76 PPIA (0.41) TAS1R3TAS1R1TAS1R2
SCHEMBL8035584 0.75 LRRK2 (0.36) SMYD3TAS1R3TAS1R1TAS1R2SLC6A2
SCHEMBL8028359 0.74 SMN1; SMN2 (0.35) TAS1R3TAS1R1TAS1R2
SCHEMBL8037250 0.74 TAS1R3 (0.45) TAS1R3TAS1R1TAS1R2
SCHEMBL8037862 0.73 CYP3A4 (0.38) CYP3A4DCUN1D1COMT
SCHEMBL8040243 0.72 PPIA (0.47)
SCHEMBL8035603 0.72 RAB9A (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009081892-A1 NOVEL CATECHOL DERIVATIVE, PHARMACEUTICAL COMPOSITION CONTAINING THE SAME, AND USE OF THOSE KISSEI PHARMACEUTICAL CO., LTD. (JP) 2009-07-02 WO disclosed