SCHEMBL8041981

SCHEMBL8041981

CCn1nnc(Sc2nc3ccccc3s2)n1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FBP1 P09467 2/20 0.50
MAPK1 P28482 5/20 0.48
CYP1A2 P05177 4/20 0.48
CYP2D6 P10635 3/20 0.48
CYP2C19 P33261 3/20 0.48
L3MBTL1 Q9Y468 2/20 0.48
CYP3A4 P08684 2/20 0.48
HIF1A Q16665 1/20 0.48
ALDH1A1 P00352 8/20 0.47
HPGD P15428 6/20 0.47
HSD17B10 Q99714 5/20 0.47
TDP1 Q9NUW8 2/20 0.47
ADRA2A P08913 1/20 0.47
ADORA3 P0DMS8 1/20 0.47
DRD2 P14416 1/20 0.47
ALOX15 P16050 1/20 0.47
ADRA2B P18089 1/20 0.47
ADRA2C P18825 1/20 0.47
DRD1 P21728 1/20 0.47
MC5R P33032 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8045191 0.90 FBP1 (0.48) FBP1MAPK1CYP1A2CYP2D6CYP2C19
SCHEMBL8046519 0.87 HSP90AA1 (0.49) FBP1MAPK1CYP1A2CYP2D6CYP2C19
SCHEMBL8052354 0.84 L3MBTL1 (0.46) FBP1MAPK1CYP1A2CYP2D6CYP2C19
SCHEMBL8043551 0.82 SMN1; SMN2 (0.51) FBP1MAPK1CYP1A2CYP2D6CYP2C19
SCHEMBL8048727 0.82 CYP1A2 (0.43) FBP1MAPK1CYP1A2CYP2D6CYP2C19
SCHEMBL8042675 0.82 ALDH1A1 (0.51) FBP1MAPK1CYP1A2CYP2D6CYP2C19
SCHEMBL8033176 0.81 HSP90AA1 (0.44) MAPK1ALDH1A1HPGDTDP1MAPT
SCHEMBL8050844 0.81 ALDH1A1 (0.47) FBP1MAPK1CYP1A2CYP2D6CYP2C19
SCHEMBL8045375 0.80 NFKB1 (0.45) ALDH1A1HPGDTDP1MAPTLMNA
SCHEMBL8041873 0.80 SMN1; SMN2 (0.45) ALDH1A1HPGDHSD17B10MAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed