SCHEMBL8043763

SCHEMBL8043763

FC(F)(F)c1cc(-c2csc(Sc3nnnn3Cc3cccs3)n2)cc(C(F)(F)F)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.40
NPSR1 Q6W5P4 3/20 0.40
USP2 O75604 2/20 0.40
OPRK1 P41145 1/20 0.36
POLB P06746 1/20 0.35
LMNA P02545 4/20 0.35
TSHR P16473 3/20 0.35
MAPK1 P28482 2/20 0.35
MAPT P10636 4/20 0.34
KDM4E B2RXH2 3/20 0.34
SMN1; SMN2 Q16637 3/20 0.34
L3MBTL1 Q9Y468 3/20 0.34
HPGD P15428 1/20 0.34
ATM Q13315 1/20 0.34
TLR8 Q9NR97 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
AR P10275 1/20 0.33
CXCR3 P49682 1/20 0.33
MAPK14 Q16539 1/20 0.33
LRRK2 Q5S007 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8045085 0.86 POLB (0.43) ALDH1A1NPSR1USP2POLBLMNA
SCHEMBL8050306 0.84 LMNA (0.41) ALDH1A1NPSR1POLBLMNATSHR
SCHEMBL8044497 0.83 HTT (0.33) ALDH1A1OPRK1POLBMAPTKDM4E
SCHEMBL8032734 0.82 ALDH1A1 (0.37) ALDH1A1NPSR1USP2POLBMAPT
SCHEMBL8045832 0.82 LMNA (0.42) ALDH1A1OPRK1POLBLMNATSHR
SCHEMBL8044430 0.81 CTSS (0.34) ALDH1A1POLBLMNAMAPTKDM4E
SCHEMBL8037022 0.80 HTT (0.38) ALDH1A1NPSR1POLBLMNAMAPT
SCHEMBL8713674 0.79 LMNA (0.40) ALDH1A1USP2LMNATSHRMAPK1
SCHEMBL8048771 0.79 MAPT (0.37) ALDH1A1LMNAMAPK1MAPTKDM4E
SCHEMBL8043192 0.79 ALDH1A1 (0.35) ALDH1A1USP2POLBLMNATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed