SCHEMBL8044646

SCHEMBL8044646

CCCn1nnnc1Sc1nc(-c2ccc(Cl)cc2)cs1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.52
LMNA P02545 5/20 0.42
MEN1 O00255 4/20 0.42
KMT2A Q03164 4/20 0.42
MAPT P10636 4/20 0.42
RAB9A P51151 3/20 0.42
NPC1 O15118 2/20 0.42
ALOX15 P16050 1/20 0.42
ALOX12 P18054 1/20 0.42
HSD17B10 Q99714 1/20 0.42
CYP1A2 P05177 4/20 0.41
CYP2C19 P33261 3/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 2/20 0.40
SREBF2 Q12772 1/20 0.39
POLB P06746 3/20 0.39
GAA P10253 1/20 0.39
HPGD P15428 1/20 0.39
KDM4E B2RXH2 2/20 0.38
ATM Q13315 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8046481 0.93 ALDH1A1 (0.44) ALDH1A1LMNAMEN1KMT2AMAPT
SCHEMBL8043207 0.91 MAPT (0.44) ALDH1A1LMNAMEN1KMT2AMAPT
SCHEMBL8034187 0.88 HTR1A (0.44) ALDH1A1LMNAMEN1KMT2AMAPT
SCHEMBL8032462 0.86 CYP2C19 (0.39) ALDH1A1LMNAMEN1KMT2AMAPT
SCHEMBL8042704 0.86 DCUN1D1 (0.44) ALDH1A1LMNAMEN1KMT2AMAPT
SCHEMBL8042146 0.84 KDM4E (0.42) LMNAMEN1KMT2AMAPTRAB9A
SCHEMBL8050040 0.84 HTT (0.51) ALDH1A1LMNAMEN1KMT2AMAPT
SCHEMBL8046147 0.83 ALDH1A1 (0.42) ALDH1A1LMNAMEN1KMT2AMAPT
SCHEMBL8720492 0.82 RAB9A (0.41) ALDH1A1LMNAMEN1KMT2ARAB9A
SCHEMBL8051108 0.82 KMT2A (0.38) ALDH1A1LMNAMEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed