SCHEMBL8046481

SCHEMBL8046481

CCCCn1nnnc1Sc1nc(-c2ccc(Cl)cc2)cs1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.44
POLB P06746 2/20 0.43
MEN1 O00255 5/20 0.42
KMT2A Q03164 5/20 0.42
CYP1A2 P05177 3/20 0.42
CYP2C19 P33261 3/20 0.42
CYP3A4 P08684 2/20 0.42
CYP2D6 P10635 1/20 0.42
PKM P14618 1/20 0.42
LMNA P02545 4/20 0.41
MAPT P10636 3/20 0.41
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
ALOX15 P16050 1/20 0.41
ALOX12 P18054 1/20 0.41
HSD17B10 Q99714 1/20 0.41
CYP2C9 P11712 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
CTDSP1 Q9GZU7 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8044646 0.93 ALDH1A1 (0.52) ALDH1A1POLBMEN1KMT2ACYP1A2
SCHEMBL8033580 0.89 POLB (0.44) ALDH1A1POLBMEN1KMT2ALMNA
SCHEMBL8043207 0.89 MAPT (0.44) ALDH1A1POLBMEN1KMT2ACYP1A2
SCHEMBL8032462 0.88 CYP2C19 (0.39) ALDH1A1MEN1KMT2ACYP1A2CYP2C19
SCHEMBL8042704 0.88 DCUN1D1 (0.44) ALDH1A1POLBMEN1KMT2ACYP1A2
SCHEMBL8720492 0.85 RAB9A (0.41) ALDH1A1MEN1KMT2ACYP1A2CYP2C19
SCHEMBL8051108 0.85 KMT2A (0.38) ALDH1A1POLBMEN1KMT2ACYP1A2
SCHEMBL8042146 0.83 KDM4E (0.42) MEN1KMT2ACYP1A2CYP2C19CYP3A4
SCHEMBL8050040 0.82 HTT (0.51) ALDH1A1MEN1KMT2ACYP1A2CYP2C19
SCHEMBL8034187 0.81 HTR1A (0.44) ALDH1A1MEN1KMT2ACYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed