SCHEMBL8046405

SCHEMBL8046405

CCOC(=O)CCCCCC(C#N)(c1ccc(OCC(F)(F)F)cc1)c1ccc(OCC(F)(F)F)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.51
NPC1 O15118 1/20 0.51
RAB9A P51151 1/20 0.51
PDK2 Q15119 2/20 0.39
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
CYP1A1 P04798 1/20 0.38
CYP1B1 Q16678 1/20 0.38
LMNA P02545 1/20 0.38
PAX8 Q06710 1/20 0.38
MAOB P27338 1/20 0.38
LTA4H P09960 2/20 0.37
MAPT P10636 1/20 0.37
BRD4 O60885 1/20 0.36
BRCA1 P38398 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
KDM4E B2RXH2 1/20 0.35
GLA P06280 1/20 0.35
FFAR1 O14842 1/20 0.35
PPARA Q07869 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8046393 0.90 L3MBTL1 (0.44) SMN1; SMN2NPC1CYP1A1CYP1B1MAOB
SCHEMBL8045896 0.85 CCR1 (0.41) SMN1; SMN2KMT2AMAPTBRD4L3MBTL1
SCHEMBL8046467 0.85 CCR1 (0.41) SMN1; SMN2KMT2AMAPTBRD4L3MBTL1
SCHEMBL8053206 0.84 FAAH (0.44) NPC1MEN1KMT2ALMNAMAPT
SCHEMBL8046383 0.84 CYP4F2 (0.40) SMN1; SMN2KDM4E
SCHEMBL8035567 0.83 CA12 (0.40) KMT2AMAOB
SCHEMBL8049639 0.82 HDAC1 (0.48) KDM4E
SCHEMBL8044912 0.82 POLB (0.36) SMN1; SMN2PDK2KMT2ALTA4HMAPT
SCHEMBL8049892 0.81 OPRM1 (0.48) SMN1; SMN2
SCHEMBL8044856 0.81 OPRM1 (0.48) SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0749957-B1 Aromatic hydroxamic acid compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2000-04-26 EP disclosed
US-5891916-A ANTINEUROGEGERATIVE AGENT TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1999-04-06 US disclosed
EP-0749957-A1 Aromatic hydroxamic acid compounds, their production and use Takeda Chemical Industries, Ltd. (JP) 1996-12-27 EP disclosed