SCHEMBL8046545

SCHEMBL8046545

S=C1N=NC(c2ccc(Br)cc2Br)=N1

nearest known ligand 0.33

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 1/20 0.33
HSP90AA1 P07900 1/20 0.32
TLR9 Q9NR96 1/20 0.32
S100A4 P26447 1/20 0.32
ALDH1A1 P00352 1/20 0.32
MAPK1 P28482 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8046050 0.77 ALDH1A1 (0.42) ALDH1A1MAPK1TDP1L3MBTL1
SCHEMBL8042855 0.70 ALDH1A1 (0.45) ALOX15ALDH1A1MAPK1
SCHEMBL11013516 0.70 ALOX15 (0.52) ALOX15HSP90AA1TLR9S100A4ALDH1A1
SCHEMBL8046152 0.68 CHRNB4 (0.31)
SCHEMBL8049878 0.68 ALOX5 (0.39) HSP90AA1ALDH1A1
Water SCHEMBL28487363 0.67 ALOX15 (0.50) ALOX15HSP90AA1TLR9S100A4ALDH1A1
SCHEMBL8044636 0.63
SCHEMBL8048510 0.63 MMP12 (0.33)
SCHEMBL8044837 0.63
SCHEMBL10479111 0.62 ALOX15 (0.44) ALOX15HSP90AA1TLR9S100A4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed