SCHEMBL8050262

SCHEMBL8050262

N#Cc1ccc(C(=O)c2ccc(O)c(F)c2)cc1

nearest known ligand 0.63

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
P4HB P07237 4/20 0.63
HSD17B1 P14061 3/20 0.50
HSD17B2 P37059 3/20 0.50
HSD17B14 Q9BPX1 1/20 0.49
ACHE P22303 1/20 0.49
VNN1 O95497 2/20 0.46
CA1 P00915 2/20 0.46
CA2 P00918 2/20 0.46
GAA P10253 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
SNCA P37840 1/20 0.44
KDM4E B2RXH2 1/20 0.44
LMNA P02545 1/20 0.44
HSD17B10 Q99714 1/20 0.44
CYP19A1 P11511 1/20 0.43
ESR1 P03372 1/20 0.43
ESR2 Q92731 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6748653 0.84 SIRT1 (0.54) P4HBHSD17B14CA1CA2GAA
SCHEMBL29748711 0.84 HSD17B1 (0.59) P4HBHSD17B1HSD17B2HSD17B14ACHE
SCHEMBL27661242 0.84 HSD17B1 (0.59) P4HBHSD17B1HSD17B2HSD17B14ACHE
SCHEMBL3433075 0.80 CA2 (0.67) P4HBVNN1CA1CA2LMNA
SCHEMBL3468841 0.79 KDM4E (0.68) P4HBHSD17B1HSD17B2ACHEVNN1
SCHEMBL9428615 0.79 ACHE (0.66) P4HBHSD17B1HSD17B2HSD17B14ACHE
SCHEMBL8047746 0.78 HTT (0.58) ACHEVNN1GAASMN1; SMN2LMNA
SCHEMBL7935350 0.78 VNN1 (0.60) VNN1CA1CA2SMN1; SMN2KDM4E
SCHEMBL200168 0.78 P4HB (0.51) P4HBHSD17B14CA2CYP19A1ESR1
SCHEMBL29826346 0.78 P4HB (0.51) P4HBHSD17B14CA2CYP19A1ESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1087934-C Use of phenalkylamines HOFFMANN LA ROCHE (CH) 2002-07-24 CN disclosed
EP-0636367-B1 Use of phenylalkylamines for producing cholesterol lowering agents HOFFMANN LA ROCHE (CH) 2000-03-29 EP disclosed
US-5637771-A Compound useful for lowering cholesterol HOFFMANN-LA ROCHE INC. (US) 1997-06-10 US disclosed
US-5574071-A ADMINISTERING PHENYLALKYLAMINO KETONES HOFFMANN-LA ROCHE INC. (US) 1996-11-12 US disclosed
US-5495048-A ANTICHOLESTEROL AGENTS HOFFMANN-LA ROCHE INC. (US) 1996-02-27 US disclosed
CN-1103781-A Use of phenalkylamines HOFFMANN LA ROCHE (CH) 1995-06-21 CN disclosed
EP-0636367-A1 Use of phenylalkylamines for producing cholesterol lowering agents F. HOFFMANN-LA ROCHE AG (CH) 1995-02-01 EP disclosed