SCHEMBL8056464

SCHEMBL8056464

COC(=O)c1cc2c(cc1C)C(c1ccccc1)=CS2(=O)=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.42
ALDH1A1 P00352 3/20 0.42
MEN1 O00255 2/20 0.42
MAPT P10636 2/20 0.42
KMT2A Q03164 2/20 0.42
GAA P10253 2/20 0.42
EGFR P00533 1/20 0.42
PTGS2 P35354 1/20 0.41
GABRA1 P14867 1/20 0.40
GABRG2 P18507 1/20 0.40
GABRB3 P28472 1/20 0.40
GABRA3 P34903 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.39
TP53 P04637 1/20 0.39
KDM4E B2RXH2 4/20 0.39
PDCD1 Q15116 1/20 0.39
CD274 Q9NZQ7 1/20 0.39
SLC6A3 Q01959 2/20 0.38
PKLR P30613 1/20 0.38
TSHR P16473 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8045188 0.85 EGFR (0.51) HPGDALDH1A1MEN1MAPTKMT2A
SCHEMBL8060790 0.85 ALDH1A1 (0.40) HPGDALDH1A1MEN1MAPTKMT2A
SCHEMBL8068448 0.74 GABRA1 (0.49) HPGDALDH1A1MEN1MAPTKMT2A
SCHEMBL8071055 0.72 ALDH1A1 (0.51) HPGDALDH1A1MEN1MAPTKMT2A
SCHEMBL8060750 0.70 LMNA (0.36) HPGDALDH1A1MEN1MAPTKMT2A
SCHEMBL3748237 0.70 EGFR (0.63) HPGDALDH1A1MEN1MAPTKMT2A
SCHEMBL16419694 0.70 GABRA1 (0.55) HPGDALDH1A1MEN1MAPTKMT2A
SCHEMBL10058712 0.70 EGFR (0.63) HPGDALDH1A1MEN1MAPTKMT2A
SCHEMBL8059705 0.69 CFTR (0.53) HPGDALDH1A1MEN1MAPTKMT2A
SCHEMBL8608047 0.69 PTGS2 (0.52) HPGDALDH1A1MEN1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6028069-A Heterocyclyl-condensed benzoylguanidines, their production and use as inhibitors of the cellular Na+/H+-antiporter MERCK PATENT GESELLSCHAFT MIT BERSCHRANKER HAFTUNG (DE) 2000-02-22 US disclosed