SCHEMBL8060790

SCHEMBL8060790

CCc1cc2c(cc1C(=O)OC)S(=O)(=O)C=C2c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.40
HPGD P15428 3/20 0.40
KMT2A Q03164 3/20 0.40
MAPT P10636 3/20 0.40
MEN1 O00255 2/20 0.40
GAA P10253 2/20 0.40
GABRA1 P14867 1/20 0.38
GABRG2 P18507 1/20 0.38
GABRB3 P28472 1/20 0.38
GABRA3 P34903 1/20 0.38
EGFR P00533 1/20 0.38
KDM4E B2RXH2 3/20 0.38
HTT P42858 1/20 0.38
LMNA P02545 1/20 0.37
PTGS2 P35354 1/20 0.37
SLC6A3 Q01959 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8056464 0.85 HPGD (0.42) ALDH1A1HPGDKMT2AMAPTMEN1
SCHEMBL8045188 0.81 EGFR (0.51) ALDH1A1HPGDKMT2AMAPTMEN1
SCHEMBL8062754 0.80 SLC9A1 (0.38)
SCHEMBL8058137 0.79 ALDH1A1 (0.36) ALDH1A1HPGDKMT2AMAPTGAA
SCHEMBL12165945 0.75 GABRA1 (0.47) ALDH1A1HPGDKMT2AMAPTMEN1
SCHEMBL12165908 0.74 KDM4E (0.50) ALDH1A1HPGDKMT2AMAPTMEN1
SCHEMBL8608965 0.71 PTGS2 (0.47) ALDH1A1HPGDKMT2AMAPTMEN1
SCHEMBL8057996 0.71 ALDH1A1 (0.37) ALDH1A1HPGDKMT2AMAPTMEN1
SCHEMBL8611218 0.70 CA2 (0.54) ALDH1A1HPGDKMT2AMAPTMEN1
SCHEMBL38659968 0.70 SLC6A3 (0.46) ALDH1A1HPGDKMT2AMAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6028069-A Heterocyclyl-condensed benzoylguanidines, their production and use as inhibitors of the cellular Na+/H+-antiporter MERCK PATENT GESELLSCHAFT MIT BERSCHRANKER HAFTUNG (DE) 2000-02-22 US disclosed