SCHEMBL8059368

SCHEMBL8059368

CN(C)c1cc(Oc2ccc(S(=O)(=O)NC(=N)N)cc2)c(S(C)(=O)=O)cc1C(=O)NC(=N)N

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 1/20 0.38
MRGPRX1 Q96LB2 2/20 0.36
MCL1 Q07820 3/20 0.35
BCL2L1 Q07817 2/20 0.35
TARS1 P26639 1/20 0.34
FLT1 P17948 3/20 0.32
FLT4 P35916 3/20 0.32
KDR P35968 3/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8068785 0.89 ALDH1A1 (0.40) SCN9A
SCHEMBL8059561 0.87 MRGPRX1 (0.41) SCN9AMRGPRX1MCL1BCL2L1TARS1
SCHEMBL8070524 0.86 FLT1 (0.42) SCN9AMCL1BCL2L1FLT1FLT4
SCHEMBL8070496 0.79 MRGPRX1 (0.43) MRGPRX1TARS1
SCHEMBL8068547 0.78 LMNA (0.41) SCN9A
SCHEMBL8059376 0.78 SCN9A (0.44) SCN9A
SCHEMBL8073839 0.72 MRGPRX1 (0.40) SCN9AMRGPRX1FLT1FLT4KDR
Hydrochloric Acid SCHEMBL8073473 0.72 THRA (0.36)
SCHEMBL8068459 0.72 SCN9A (0.36) SCN9A
SCHEMBL8446348 0.70 CA2 (0.43) MRGPRX1CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6057322-A USEFUL IN TREATMENT OF CARDIOVASCULAR DISEASES HOECHST AKTIENGESELLSCHAFT (DE) 2000-05-02 US disclosed