SCHEMBL8066342

SCHEMBL8066342

COc1ccc(N(C(=O)Oc2c3ccccc3nc3ccccc23)S(=O)(=O)c2ccc(CCC(=O)ON3C(=O)CCC3=O)cc2)c(OC)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.38
KEAP1 Q14145 5/20 0.37
PIK3CG P48736 1/20 0.37
CA2 P00918 5/20 0.36
CA12 O43570 2/20 0.36
CA1 P00915 2/20 0.36
CA9 Q16790 2/20 0.36
LMNA P02545 2/20 0.36
GAA P10253 1/20 0.36
PKM P14618 1/20 0.36
HTT P42858 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
USP2 O75604 1/20 0.35
HPGD P15428 1/20 0.35
ALOX15 P16050 1/20 0.35
TSHR P16473 1/20 0.35
NFE2L2 Q16236 4/20 0.35
KMT2A Q03164 2/20 0.35
MEN1 O00255 1/20 0.35
POLB P06746 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8469817 0.90 KEAP1 (0.40) ALDH1A1KEAP1PIK3CGCA2CA12
SCHEMBL8074300 0.89 ALDH1A1 (0.40) ALDH1A1KEAP1PIK3CGCA2LMNA
Bromide SCHEMBL8080918 0.86 KEAP1 (0.45) ALDH1A1KEAP1CA2CA12CA1
SCHEMBL8076290 0.86 KEAP1 (0.40) KEAP1PIK3CGCA2CA12CA1
SCHEMBL8079548 0.84 ALDH1A1 (0.38) ALDH1A1KEAP1CA2LMNAGAA
SCHEMBL8079566 0.83 LMNA (0.37) ALDH1A1CA2CA12CA1CA9
SCHEMBL9407932 0.80 LMNA (0.35) ALDH1A1CA2CA12CA1CA9
SCHEMBL8470105 0.80 ALDH1A1 (0.43) ALDH1A1KEAP1PIK3CGLMNAGAA
SCHEMBL9407920 0.80 CXCR3 (0.34) CA2LMNASMN1; SMN2MAPT
SCHEMBL8074297 0.80 TSHR (0.40) ALDH1A1KEAP1CA2CA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0330050-B1 Special chemiluminescent acridine derivatives and their use in luminescence immunoassays DADE BEHRING MARBURG GMBH (DE) 2000-08-23 EP disclosed
EP-0602524-A1 Chemiluminescence marked sequences and their use in sequence testing HOECHST AKTIENGESELLSCHAFT (DE) 1994-06-22 EP disclosed
EP-0330050-A2 Special chemiluminescent acridine derivatives and their use in luminescence immunoassays HOECHST AKTIENGESELLSCHAFT (DE) 1989-08-30 EP disclosed