Piperidine

Piperidine

SCHEMBL8068938

C1CCNCC1.CCNS(=O)(=O)c1ccc(Oc2ccc(C(=O)O)cc2S(C)(=O)=O)cc1

nearest known ligand 0.42

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.42
ALDH1A1 P00352 4/20 0.40
NPSR1 Q6W5P4 2/20 0.40
MAPT P10636 2/20 0.40
GAA P10253 1/20 0.40
KMT2A Q03164 1/20 0.39
GFER P55789 1/20 0.38
POLB P06746 1/20 0.37
PKM P14618 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
MEP1B Q16820 2/20 0.37
CCR1 P32246 1/20 0.37
CCR2 P41597 1/20 0.37
CCR5 P51681 1/20 0.37
LMNA P02545 1/20 0.36
ADAMTS4 O75173 1/20 0.36
MMP1 P03956 1/20 0.36
MMP2 P08253 1/20 0.36
MMP13 P45452 1/20 0.36
MMP14 P50281 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8068934 0.80 SIGMAR1 (0.51) MAPTGAAKMT2APOLBCCR2
SCHEMBL8068849 0.78 ALDH1A1 (0.54) TSHRALDH1A1MAPTKMT2AGFER
SCHEMBL8059681 0.77 TTR (0.45) NPSR1MAPTGAAGFERPOLB
SCHEMBL8073502 0.76 TTR (0.51) ALDH1A1NPSR1MAPTGAAPOLB
SCHEMBL8073771 0.75 KMT2A (0.58) TSHRALDH1A1NPSR1KMT2APOLB
Piperidine SCHEMBL8073727 0.74 PKM (0.48) TSHRALDH1A1NPSR1POLBPKM
SCHEMBL8447165 0.74 NPSR1 (0.45) ALDH1A1NPSR1GFERPOLBPKM
SCHEMBL8059364 0.74 PKM (0.55) ALDH1A1POLBPKMTDP1L3MBTL1
SCHEMBL8070556 0.74 MAPT (0.47) TSHRMAPTKMT2APOLBPKM
SCHEMBL8059678 0.74 NPSR1 (0.44) ALDH1A1NPSR1KMT2APOLBPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6057322-A USEFUL IN TREATMENT OF CARDIOVASCULAR DISEASES HOECHST AKTIENGESELLSCHAFT (DE) 2000-05-02 US disclosed