SCHEMBL8068950

SCHEMBL8068950

CN(C)CCc1ccc(Oc2ccc(C(=O)O)cc2C(F)(F)F)c(C=S)c1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
THRA P10827 2/20 0.43
THRB P10828 2/20 0.43
RXRA P19793 3/20 0.41
RXRB P28702 3/20 0.41
RXRG P48443 3/20 0.41
LPAR1 Q92633 1/20 0.41
LPAR5 Q9H1C0 1/20 0.41
MRGPRX4 Q96LA9 6/20 0.37
SIRT1 Q96EB6 1/20 0.37
ROCK2 O75116 1/20 0.35
POLB P06746 1/20 0.35
PKM P14618 1/20 0.35
SRD5A2 P31213 1/20 0.34
BCHE P06276 1/20 0.34
ACHE P22303 1/20 0.34
S1PR1 P21453 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8068641 0.84 SIRT1 (0.41) THRATHRBLPAR1LPAR5MRGPRX4
Hydrochloric Acid SCHEMBL8073699 0.81 PKM (0.43) THRATHRBPOLBPKMBCHE
SCHEMBL8068627 0.72 LPAR1 (0.48) THRATHRBLPAR1LPAR5MRGPRX4
SCHEMBL8068951 0.72 LPAR1 (0.46) THRATHRBRXRARXRBRXRG
SCHEMBL8059726 0.69 THRA (0.47) THRATHRBRXRARXRBRXRG
SCHEMBL8074970 0.68 SLC6A2 (0.45) THRATHRBLPAR1LPAR5SIRT1
Hydrochloric Acid SCHEMBL8070331 0.67 SLC6A2 (0.44) THRATHRBLPAR1LPAR5SIRT1
SCHEMBL30835355 0.67 RXRA (0.46) THRATHRBRXRARXRBRXRG
SCHEMBL615379 0.66 CA12 (0.62) RXRARXRBRXRGMRGPRX4PKM
SCHEMBL3529077 0.66 HCAR3 (0.46) THRATHRBRXRARXRBRXRG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6057322-A USEFUL IN TREATMENT OF CARDIOVASCULAR DISEASES HOECHST AKTIENGESELLSCHAFT (DE) 2000-05-02 US disclosed