SCHEMBL8078749

SCHEMBL8078749

CC(C)(C)Oc1cccc(-c2cccc(S)c2-c2cccc(OC(C)(C)C)c2)c1.Cc1ccc(S(=O)(=O)O)cc1

nearest known ligand 0.36

Known targets — ChEMBL curated mechanism

ABL1BMXBRAFBTKCHRNA4CHRNB2CSNK1EEGFRERBB2F10FLT1FLT3FLT4IGF1RINSRITKJAK3KDRKITOPRM1PARP1PARP2PDGFRBPIK3CDRAF1RETSLC18A2TECTXKdacAdacBdacCftsImrcAmrcBmrdArplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 1/20 0.36
PRKDC P78527 1/20 0.36
ALDH1A1 P00352 4/20 0.35
TDP1 Q9NUW8 3/20 0.35
KDM4E B2RXH2 3/20 0.35
HTT P42858 2/20 0.35
L3MBTL1 Q9Y468 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
MAPT P10636 2/20 0.35
LMNA P02545 1/20 0.35
PTGES2 Q9H7Z7 1/20 0.34
ALKBH3 Q96Q83 1/20 0.34
SNCA P37840 1/20 0.33
SCN9A Q15858 1/20 0.33
CYP2D6 P10635 2/20 0.33
MAPK1 P28482 1/20 0.33
MEN1 O00255 4/20 0.32
KMT2A Q03164 4/20 0.32
ACLY P53396 1/20 0.32
TP53 P04637 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8644650 0.90 PRKDC (0.35) PRKDCMAPTSCN9ACYP2D6TP53
SCHEMBL219087 0.87 TDP1 (0.36) ALDH1A1TDP1KDM4EHTTL3MBTL1
SCHEMBL244495 0.83 KDM4E (0.40) PRKDCALDH1A1KDM4EMEN1KMT2A
SCHEMBL8645387 0.80 AKR1C3 (0.38) PRKDCSCN9ANR1H2NR1H3AKR1C4
SCHEMBL3144542 0.78 LMNA (0.44) ALDH1A1TDP1KDM4EHTTL3MBTL1
SCHEMBL3140909 0.76 LMNA (0.42) ALDH1A1TDP1KDM4EHTTL3MBTL1
SCHEMBL3143806 0.76 PTGS2 (0.42) ALDH1A1TDP1KDM4EHTTL3MBTL1
SCHEMBL3135090 0.74 LMNA (0.45) ALDH1A1TDP1KDM4EHTTL3MBTL1
SCHEMBL8647456 0.74 FABP4 (0.35) MAPTNR1H2NR1H3AKR1C3AKR1C2
SCHEMBL3132925 0.74 ALDH1A1 (0.42) ALDH1A1TDP1KDM4EHTTL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6106993-A HIGHLY SENSITIVE TO ACTINIC RADIATION SUCH AS DEEP-UV, ELECTRON BEAM AND X-RAY, CAN BE DEVELOPED WITH ALKALINE AQUEOUS SOLUTION TO FORM A PATTERN, AND IS THUS SUITABLE FOR USE IN A FINE PATTERNING TECHNIQUE SHIN-ETSU CHEMICAL CO., LTD. (JP) 2000-08-22 US disclosed