SCHEMBL808039

SCHEMBL808039

C=C(/N=C(N)\N=C(/N)c1noc(N2CCC(NC(=O)C(F)(F)F)CC2)n1)N(C)c1ccccc1

nearest known ligand 0.33

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CKS1B P61024 1/20 0.33
SKP1 P63208 1/20 0.33
SKP2 Q13309 1/20 0.33
BTK Q06187 3/20 0.33
SMO Q99835 2/20 0.33
POLB P06746 1/20 0.33
PKM P14618 1/20 0.32
DRD2 P14416 3/20 0.32
HTR2A P28223 3/20 0.32
DRD3 P35462 3/20 0.32
HTR1A P08908 2/20 0.32
SSTR4 P31391 1/20 0.31
HDAC4 P56524 2/20 0.31
HDAC6 Q9UBN7 2/20 0.31
SMPD3 Q9NY59 1/20 0.31
HDAC8 Q9BY41 1/20 0.31
CYP2C9 P11712 1/20 0.31
EPHX2 P34913 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL808032 0.83 DHFR (0.34) POLBDRD2
SCHEMBL808024 0.81 TSHR (0.37)
SCHEMBL808232 0.80 CNR2 (0.32) POLB
SCHEMBL808046 0.79 GAA (0.31) HDAC4HDAC6HDAC8
SCHEMBL808343 0.77 SCD (0.34)
SCHEMBL808329 0.75 SCD (0.38)
SCHEMBL808026 0.74
SCHEMBL808236 0.72 TSHR (0.39) PKMHDAC6HDAC8
SCHEMBL807935 0.71 SMN1; SMN2 (0.41) SMOHDAC6HDAC8CYP2C9EPHX2
SCHEMBL796294 0.71 SMO (0.39) CKS1BSKP1SKP2SMOPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012035023-A1 TRIAZINE-OXADIAZOLES NOVARTIS AG (CH) 2012-03-22 WO disclosed