SCHEMBL808223

SCHEMBL808223

C=C(/N=C(N)\N=C(/N)c1noc(C2CCN(S(=O)(=O)CC)CC2)n1)N(C)c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.43
RAB9A P51151 3/20 0.43
HTT P42858 2/20 0.43
NPC1 O15118 2/20 0.43
GAA P10253 4/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
KMT2A Q03164 3/20 0.39
ALDH1A1 P00352 2/20 0.39
MAPT P10636 2/20 0.39
MEN1 O00255 2/20 0.39
CYP2C9 P11712 1/20 0.39
APEX1 P27695 1/20 0.39
HSD17B10 Q99714 2/20 0.39
TSHR P16473 1/20 0.39
HPGD P15428 3/20 0.36
KDM4E B2RXH2 1/20 0.36
ADRB2 P07550 1/20 0.36
GFER P55789 2/20 0.34
MAPK1 P28482 1/20 0.34
TUBB4A P04350 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL808048 0.93 LMNA (0.36) LMNARAB9AHTTNPC1GAA
SCHEMBL10286918 0.92 GAA (0.39) LMNARAB9AHTTNPC1GAA
SCHEMBL10286916 0.90 ALDH1A1 (0.38) LMNARAB9AHTTNPC1GAA
SCHEMBL808022 0.88 LMNA (0.35) LMNARAB9AHTTNPC1GAA
SCHEMBL807956 0.85 PRCP (0.35) GAAKMT2AALDH1A1MAPTMEN1
SCHEMBL807935 0.84 SMN1; SMN2 (0.41) LMNAGAASMN1; SMN2KMT2AALDH1A1
SCHEMBL10286917 0.84 GRM5 (0.41) LMNAHTTGAASMN1; SMN2KMT2A
SCHEMBL10286920 0.82 SMN1; SMN2 (0.41) GAASMN1; SMN2KMT2AMAPTMEN1
SCHEMBL10287790 0.78 LMNA (0.38) LMNARAB9AHTTNPC1GAA
SCHEMBL808032 0.77 DHFR (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012035023-A1 TRIAZINE-OXADIAZOLES NOVARTIS AG (CH) 2012-03-22 WO disclosed