SCHEMBL8083334

SCHEMBL8083334

CNC(=S)Nc1ccc(-c2nc(N)cc(C3(S(=O)(=O)c4ccc(F)cc4)CC3)n2)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.41
CA2 P00918 2/20 0.41
CA4 P22748 2/20 0.41
CA9 Q16790 2/20 0.41
ALDH1A1 P00352 4/20 0.40
PIK3CA P42336 5/20 0.37
PIK3CD O00329 3/20 0.37
MTOR P42345 2/20 0.37
PPIA P62937 1/20 0.37
PIK3CB P42338 1/20 0.37
PIK3CG P48736 1/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
PTGS2 P35354 1/20 0.36
LMNA P02545 1/20 0.36
GAA P10253 1/20 0.36
ALOX12 P18054 1/20 0.35
PIK3R1 P27986 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
KDM1A O60341 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8099045 0.91 MAPT (0.39) CA1CA2CA9ALDH1A1PIK3CA
SCHEMBL8083973 0.90 ALDH1A1 (0.43) CA1CA2CA4CA9ALDH1A1
SCHEMBL8097689 0.90 ALDH1A1 (0.40) CA1CA2CA4CA9ALDH1A1
SCHEMBL8083200 0.87 ALDH1A1 (0.43) CA1CA2CA4CA9ALDH1A1
SCHEMBL8092637 0.84 KMT2A (0.42) CA1CA2CA9PIK3CAPIK3CD
SCHEMBL8089917 0.82 PIK3CA (0.39) CA2CA9ALDH1A1PIK3CAPIK3CD
SCHEMBL8099408 0.82 CA2 (0.42) CA1CA2CA4CA9ALDH1A1
SCHEMBL8100086 0.82 PIK3CD (0.53) ALDH1A1PIK3CAPIK3CDMTORPIK3CB
SCHEMBL8098812 0.82 NPC1 (0.43) CA1CA2CA4CA9ALDH1A1
SCHEMBL8097426 0.81 NAMPT (0.41) CA1CA2CA4CA9ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007748-A2 TRISUBSTITUTED PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PROLIFERATIVE DISEASES ASTRAZENECA AB (SE) 2009-01-15 WO disclosed