SCHEMBL8097689

SCHEMBL8097689

NC(=S)Nc1ccc(-c2nc(N)cc(C3(S(=O)(=O)c4ccc(F)cc4)CC3)n2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.40
PIK3CA P42336 4/20 0.38
PIK3R1 P27986 1/20 0.38
CA2 P00918 4/20 0.38
CA1 P00915 3/20 0.38
CA4 P22748 3/20 0.38
CA9 Q16790 3/20 0.38
MTOR P42345 3/20 0.35
PIK3CG P48736 2/20 0.35
CSF1R P07333 1/20 0.35
PTPN11 Q06124 1/20 0.34
KDM1A O60341 1/20 0.34
CA7 P43166 2/20 0.34
CA12 O43570 1/20 0.34
NAMPT P43490 1/20 0.34
PIK3CD O00329 1/20 0.34
PIK3CB P42338 1/20 0.34
GAA P10253 2/20 0.33
CFTR P13569 1/20 0.33
LMNA P02545 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8083200 0.91 ALDH1A1 (0.43) ALDH1A1PIK3CAPIK3R1CA2CA1
SCHEMBL8084155 0.90 MAPT (0.39) ALDH1A1PIK3CAPIK3R1CA2CA1
SCHEMBL8083334 0.90 CA1 (0.41) ALDH1A1PIK3CAPIK3R1CA2CA1
SCHEMBL8083973 0.87 ALDH1A1 (0.43) ALDH1A1PIK3CAPIK3R1CA2CA1
SCHEMBL8098812 0.84 NPC1 (0.43) ALDH1A1CA2CA1CA4CA9
SCHEMBL8084829 0.83 ATR (0.41) ALDH1A1PIK3CAMTORPIK3CGPIK3CD
SCHEMBL8097966 0.83 KIF11 (0.37) ALDH1A1PIK3CAMTORPIK3CGNAMPT
SCHEMBL8099408 0.83 CA2 (0.42) ALDH1A1PIK3CACA2CA1CA4
SCHEMBL8090391 0.82 CA1 (0.41) ALDH1A1PIK3CACA2CA1CA4
SCHEMBL8097426 0.82 NAMPT (0.41) ALDH1A1PIK3CACA2CA1CA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007748-A2 TRISUBSTITUTED PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PROLIFERATIVE DISEASES ASTRAZENECA AB (SE) 2009-01-15 WO disclosed