SCHEMBL8083200

SCHEMBL8083200

NC(=O)Nc1ccc(-c2nc(N)cc(C3(S(=O)(=O)c4ccc(F)cc4)CC3)n2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.43
KIF11 P52732 1/20 0.40
MEN1 O00255 1/20 0.38
IKBKB O14920 1/20 0.38
JAK2 O60674 1/20 0.38
EIF2AK2 P19525 1/20 0.38
KMT2A Q03164 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
IDO1 P14902 1/20 0.38
TDO2 P48775 1/20 0.38
PIK3CA P42336 3/20 0.37
PIK3R1 P27986 1/20 0.37
CSF1R P07333 1/20 0.37
CA2 P00918 3/20 0.37
CA1 P00915 2/20 0.37
CA4 P22748 2/20 0.37
CA7 P43166 2/20 0.37
MTOR P42345 2/20 0.37
CA9 Q16790 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8097966 0.92 KIF11 (0.37) ALDH1A1KIF11MEN1IKBKBJAK2
SCHEMBL8097689 0.91 ALDH1A1 (0.40) ALDH1A1PIK3CAPIK3R1CSF1RCA2
SCHEMBL8084982 0.90 KIF11 (0.38) ALDH1A1KIF11MEN1KMT2AIDO1
SCHEMBL8091293 0.90 MAPT (0.42) ALDH1A1KIF11MEN1KMT2APIK3CA
SCHEMBL8083973 0.89 ALDH1A1 (0.43) ALDH1A1MEN1KMT2APIK3CAPIK3R1
SCHEMBL8090868 0.89 MTOR (0.38) ALDH1A1KIF11MEN1IKBKBKMT2A
SCHEMBL8091026 0.89 NAMPT (0.36) ALDH1A1KIF11MEN1IKBKBJAK2
SCHEMBL8085029 0.87 KIF11 (0.38) ALDH1A1KIF11MEN1IKBKBKMT2A
SCHEMBL8104712 0.87 IDO1 (0.40) ALDH1A1KIF11MEN1IKBKBJAK2
SCHEMBL8082685 0.87 IDO1 (0.40) ALDH1A1IDO1TDO2PIK3CAMTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007748-A2 TRISUBSTITUTED PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PROLIFERATIVE DISEASES ASTRAZENECA AB (SE) 2009-01-15 WO disclosed