SCHEMBL8083977

SCHEMBL8083977

Nc1cc(C2(SO)CC2)nc(-c2ccc(NC(=O)NCc3ncc[nH]3)cc2)n1

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
FPR2 P25090 1/20 0.52
MAPK1 P28482 1/20 0.39
ADORA3 P0DMS8 2/20 0.36
ADORA2A P29274 2/20 0.36
ADORA1 P30542 2/20 0.36
KLK1 P06870 1/20 0.36
KLK5 Q9Y337 1/20 0.36
ADORA2B P29275 1/20 0.36
PIK3CD O00329 7/20 0.36
PIK3CA P42336 3/20 0.36
ROCK2 O75116 5/20 0.35
SLC40A1 Q9NP59 1/20 0.33
NTRK1 P04629 1/20 0.33
ROCK1 Q13464 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8091600 0.82 PIK3CA (0.40) PIK3CDPIK3CA
SCHEMBL8096884 0.81 KDM4E (0.39) PIK3CDPIK3CA
SCHEMBL8092177 0.81 FPR2 (0.47) FPR2MAPK1PIK3CDROCK2ROCK1
SCHEMBL8090988 0.80 MTOR (0.44) PIK3CDPIK3CA
SCHEMBL8092577 0.80 FPR2 (0.46) FPR2MAPK1
SCHEMBL8089937 0.79 KIF11 (0.39)
SCHEMBL8083982 0.78 PIK3CD (0.34) PIK3CDPIK3CA
SCHEMBL8099890 0.78 GHSR (0.39) PIK3CDROCK2
SCHEMBL8215025 0.78 FPR2 (0.51) FPR2MAPK1ADORA3ADORA2AADORA1
SCHEMBL8095224 0.77 PIK3CD (0.34) MAPK1PIK3CDPIK3CAROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007748-A2 TRISUBSTITUTED PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PROLIFERATIVE DISEASES ASTRAZENECA AB (SE) 2009-01-15 WO disclosed