SCHEMBL8091440

SCHEMBL8091440

COc1ccc(CCc2ccc[c]c2CCCc2ccccc2)cc1

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 3/20 0.52
SIGMAR1 Q99720 3/20 0.49
TDP1 Q9NUW8 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
CALM1 P0DP23 1/20 0.45
LTA4H P09960 1/20 0.45
ALDH1A1 P00352 1/20 0.43
ALOX5 P09917 1/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
PLAAT3 P53816 1/20 0.41
PLAAT5 Q96KN8 1/20 0.41
PLAAT2 Q9NWW9 1/20 0.41
PLAAT4 Q9UL19 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7426680 0.95 SIGMAR1 (0.49) ABCB1SIGMAR1TDP1L3MBTL1CALM1
SCHEMBL6570928 0.82 HTR2A (0.42) SIGMAR1
SCHEMBL10422126 0.79 HTR1A (0.43) ABCB1TDP1ALDH1A1
SCHEMBL5632470 0.79 LTA4H (0.69) ABCB1SIGMAR1TDP1L3MBTL1CALM1
SCHEMBL5332631 0.79 KCNH2 (0.40) SIGMAR1ALDH1A1
SCHEMBL8078997 0.78 SIGMAR1 (0.49) SIGMAR1TDP1L3MBTL1CALM1LTA4H
SCHEMBL140371 0.78 ADRA1A (0.40) L3MBTL1MEN1KMT2A
SCHEMBL3365900 0.76 ABCB1 (0.47) ABCB1
SCHEMBL2355634 0.75 LTA4H (0.75) ABCB1SIGMAR1TDP1L3MBTL1LTA4H
SCHEMBL8090170 0.75 TDP1 (0.49) ABCB1SIGMAR1TDP1L3MBTL1CALM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6124328-A TREATING NERVE CELLS WITH A NEUROTROPHIC AGENT; PROMOTING REPAIR OF NEURONAL DAMAGE CAUSED BY DISEASE OR PHYSICAL TRAUMA VERTEX PHARMACEUTICALS INCORPORATED (US) 2000-09-26 US disclosed
US-6037370-A TREATING ALZHEIMER*S DISEASE, AMYOTROPHIC LATERAL SCLEROSIS, PARKINSON*S DISEASE, AND OTHER NERVOUS SYSTEM DISORDERS WITH PEPTIDE DERIVATIVES VERTEX PHARMACEUTICALS INCORPORATED (US) 2000-03-14 US disclosed