SCHEMBL8093555

SCHEMBL8093555

CSc1ccnc2c1N(C)c1cccnc1N2C

nearest known ligand 0.33

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
ADORA3 P0DMS8 1/20 0.30
ADORA2A P29274 1/20 0.30
ADORA1 P30542 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8101458 0.94 GRM5 (0.33) GRM5L3MBTL1ADORA3ADORA2AADORA1
SCHEMBL8103219 0.77 ADORA3 (0.39) ADORA3ADORA2AADORA1
SCHEMBL8093553 0.76 ADORA3 (0.31) ADORA3ADORA2AADORA1
SCHEMBL8101449 0.75 MYC (0.40) L3MBTL1ADORA3ADORA2AADORA1
SCHEMBL8101368 0.75 TRIM24 (0.39) L3MBTL1ADORA3ADORA2AADORA1
SCHEMBL8101364 0.72 KDM4E (0.40) L3MBTL1
SCHEMBL8107544 0.71 ALDH1A1 (0.33)
SCHEMBL8109284 0.71 GAA (0.37) ADORA3ADORA2AADORA1
SCHEMBL8093773 0.69 CHRM2 (0.33)
SCHEMBL8103161 0.69 KDM4E (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6127369-A 5,10-dihydrodipyrido[2,3-b:2,3-e]pyrazin and 5,10-dihydrodipyrido[2,3-b:3,2-e]pyrazin compounds ADIR ET COMPAGNIE (FR) 2000-10-03 US disclosed