SCHEMBL8103353

SCHEMBL8103353

COc1ccccc1N1CCNCC1.FC(F)(F)c1cccc(N2CCNCC2)c1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR3E A5X5Y0 2/20 0.69
HTR3B O95264 2/20 0.69
HTR3A P46098 2/20 0.69
HTR3D Q70Z44 2/20 0.69
HTR3C Q8WXA8 2/20 0.69
SIGMAR1 Q99720 2/20 0.69
ALDH1A1 P00352 1/20 0.69
HTR1D P28221 1/20 0.69
HTR2C P28335 1/20 0.69
MAPT P10636 4/20 0.67
THRB P10828 1/20 0.67
ADRB1 P08588 2/20 0.64
DRD2 P14416 2/20 0.64
HTR6 P50406 2/20 0.64
CYP2C19 P33261 1/20 0.64
DRD3 P35462 1/20 0.64
LMNA P02545 4/20 0.63
TSHR P16473 4/20 0.56
HTR7 P34969 4/20 0.56
HTR1A P08908 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6094745 0.83 ALDH1A1 (1.00) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL231692 0.83 ALDH1A1 (1.00) HTR3EHTR3BHTR3AHTR3DHTR3C
Phenylpiperazine SCHEMBL3440604 0.82 HTR3A (0.84) HTR3EHTR3BHTR3AHTR3DHTR3C
Hydrochloric Acid SCHEMBL720648 0.82 THRB (1.00) HTR3EHTR3BHTR3AHTR3DHTR3C
Bromide SCHEMBL9146763 0.82 ALDH1A1 (0.97) HTR3EHTR3BHTR3AHTR3DHTR3C
Hydrochloric Acid SCHEMBL12818335 0.82 THRB (1.00) HTR3EHTR3BHTR3AHTR3DHTR3C
Piperazine SCHEMBL28225297 0.80 THRB (0.97) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL379 0.80 HTR3A (1.00) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL29396943 0.80 HTR3A (1.00) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL6366499 0.80 HTR3A (1.00) HTR3EHTR3BHTR3AHTR3DHTR3C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0973936-A1 COMBINATORIAL LIBRARIES OF PEPTIDOMIMETIC AMINOTHIOETHER ACIDS ELI LILLY AND COMPANY (US) 2000-01-26 EP disclosed
WO-1998046786-A1 COMBINATORIAL LIBRARIES OF PEPTIDOMIMETIC AMINOTHIOETHER ACIDS ELI LILLY AND COMPANY (US) 1998-10-22 WO disclosed