SCHEMBL8103437

SCHEMBL8103437

CCCCN1c2ccc(C=O)nc2N(CCCC)c2cccnc21

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.39
MAPK1 P28482 2/20 0.35
TP53 P04637 1/20 0.35
CFTR P13569 1/20 0.33
MAPT P10636 2/20 0.33
CHRM2 P08172 1/20 0.33
ADRA2A P08913 1/20 0.33
ADRA2B P18089 1/20 0.33
ADRA2C P18825 1/20 0.33
ALDH2 P05091 1/20 0.33
ALDH3A1 P30838 1/20 0.33
CDC25A P30304 2/20 0.32
CES1 P23141 2/20 0.32
PDE4A P27815 1/20 0.32
PDE4B Q07343 1/20 0.32
PDE4C Q08493 1/20 0.32
PDE4D Q08499 1/20 0.32
PDF Q9HBH1 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2D6 P10635 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8101315 0.96 ALDH1A1 (0.38) ALDH1A1MAPK1TP53CFTRMAPT
SCHEMBL8103457 0.83 ALDH1A1 (0.44) ALDH1A1MAPK1TP53CFTRMAPT
SCHEMBL8101881 0.79 ALDH1A1 (0.43) ALDH1A1MAPK1TP53CFTRMAPT
SCHEMBL8107634 0.78 PKM (0.37) ALDH1A1MAPK1TP53CFTRMAPT
SCHEMBL8109276 0.76 ALDH1A1 (0.46) ALDH1A1BRD4
SCHEMBL8107632 0.76 ADRA2A (0.36) ALDH1A1MAPK1TP53CFTRMAPT
SCHEMBL8101460 0.74 PKM (0.36) ALDH1A1MAPK1TP53MAPTALDH2
SCHEMBL4316094 0.74 ADRA2A (0.51) MAPTADRA2AADRA2BADRA2CCYP2D6
SCHEMBL8107425 0.74 ADRA2A (0.51) MAPTADRA2AADRA2BADRA2CCYP2D6
SCHEMBL8107564 0.68 ADRA2A (0.47) ADRA2AADRA2BADRA2CCYP2D6BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6127369-A 5,10-dihydrodipyrido[2,3-b:2,3-e]pyrazin and 5,10-dihydrodipyrido[2,3-b:3,2-e]pyrazin compounds ADIR ET COMPAGNIE (FR) 2000-10-03 US disclosed