SCHEMBL8104712

SCHEMBL8104712

NC(=O)Nc1ccc(-c2nc(N)cc(C3(S(=O)(=O)c4ccc(F)cc4F)CC3)n2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.40
TDO2 P48775 2/20 0.40
ALDH1A1 P00352 1/20 0.37
PIK3CA P42336 3/20 0.36
MTOR P42345 2/20 0.36
PIK3CG P48736 1/20 0.36
NAMPT P43490 3/20 0.36
HDAC3 O15379 2/20 0.35
SGK1 O00141 5/20 0.34
MEN1 O00255 1/20 0.34
IKBKB O14920 1/20 0.34
JAK2 O60674 1/20 0.34
EIF2AK2 P19525 1/20 0.34
KMT2A Q03164 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
NCOR2 Q9Y618 1/20 0.34
KIF11 P52732 1/20 0.33
MET P08581 1/20 0.33
PIK3CD O00329 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8082685 0.93 IDO1 (0.40) IDO1TDO2ALDH1A1PIK3CAMTOR
SCHEMBL8083416 0.90 PIK3R1 (0.39) IDO1TDO2ALDH1A1PIK3CANAMPT
SCHEMBL8084965 0.89 IDO1 (0.39) IDO1TDO2ALDH1A1PIK3CAMTOR
SCHEMBL8083200 0.87 ALDH1A1 (0.43) IDO1TDO2ALDH1A1PIK3CAMTOR
SCHEMBL8084961 0.87 NAMPT (0.41) PIK3CAMTORPIK3CGNAMPTHDAC3
SCHEMBL8100133 0.87 NAMPT (0.41) PIK3CAMTORPIK3CGNAMPTHDAC3
SCHEMBL8093534 0.86 NAMPT (0.41) PIK3CAMTORPIK3CGNAMPTHDAC3
SCHEMBL8097966 0.85 KIF11 (0.37) IDO1TDO2ALDH1A1PIK3CAMTOR
SCHEMBL8090834 0.85 KIF11 (0.35) IDO1TDO2ALDH1A1MEN1IKBKB
SCHEMBL8084982 0.84 KIF11 (0.38) IDO1TDO2ALDH1A1NAMPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007748-A2 TRISUBSTITUTED PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PROLIFERATIVE DISEASES ASTRAZENECA AB (SE) 2009-01-15 WO disclosed