SCHEMBL8090834

SCHEMBL8090834

NC(=O)Nc1ccc(-c2nc(N)cc(C3(S(=O)(=O)c4c(F)cccc4F)CC3)n2)cc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 5/20 0.35
KDR P35968 2/20 0.34
EPHB4 P54760 1/20 0.34
TEK Q02763 1/20 0.34
ALDH1A1 P00352 2/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
KIT P10721 1/20 0.33
FLT3 P36888 1/20 0.33
IDO1 P14902 1/20 0.33
TDO2 P48775 1/20 0.33
IKBKB O14920 1/20 0.33
JAK2 O60674 1/20 0.33
EIF2AK2 P19525 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
RORC P51449 2/20 0.33
MET P08581 1/20 0.33
PKM P14618 1/20 0.32
HDAC1 Q13547 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8083416 0.89 PIK3R1 (0.39) KIF11ALDH1A1MEN1KMT2AIDO1
SCHEMBL8090837 0.86 MTOR (0.38) PIK3CDCA1CA2MAPT
SCHEMBL8097253 0.86 PIK3CD (0.36) MEN1KMT2APIK3CDMAPT
SCHEMBL8084982 0.85 KIF11 (0.38) KIF11KDREPHB4TEKALDH1A1
SCHEMBL8083200 0.85 ALDH1A1 (0.43) KIF11ALDH1A1MEN1KMT2AIDO1
SCHEMBL8097966 0.85 KIF11 (0.37) KIF11ALDH1A1MEN1KMT2AIDO1
SCHEMBL8091293 0.85 MAPT (0.42) KIF11ALDH1A1MEN1KMT2ACA1
SCHEMBL8104712 0.85 IDO1 (0.40) KIF11ALDH1A1MEN1KMT2AIDO1
SCHEMBL8082685 0.85 IDO1 (0.40) ALDH1A1IDO1TDO2
SCHEMBL8083616 0.82 ATR (0.42) KIF11ALDH1A1MEN1KMT2APIK3CD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007748-A2 TRISUBSTITUTED PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PROLIFERATIVE DISEASES ASTRAZENECA AB (SE) 2009-01-15 WO disclosed