SCHEMBL8082685

SCHEMBL8082685

NC(=O)Nc1ccc(-c2nc(N)cc(C3(S(=O)(=O)c4cc(F)ccc4F)CC3)n2)cc1

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.40
TDO2 P48775 2/20 0.40
SGK1 O00141 15/20 0.39
ALDH1A1 P00352 1/20 0.37
PIK3CA P42336 2/20 0.35
HDAC3 O15379 1/20 0.35
MTOR P42345 1/20 0.35
PIK3CG P48736 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8104712 0.93 IDO1 (0.40) IDO1TDO2SGK1ALDH1A1PIK3CA
SCHEMBL8084965 0.91 IDO1 (0.39) IDO1TDO2SGK1ALDH1A1PIK3CA
SCHEMBL8083416 0.90 PIK3R1 (0.39) IDO1TDO2SGK1ALDH1A1PIK3CA
SCHEMBL8083200 0.87 ALDH1A1 (0.43) IDO1TDO2ALDH1A1PIK3CAMTOR
SCHEMBL8090580 0.87 NAMPT (0.39) SGK1PIK3CAHDAC3MTORPIK3CG
SCHEMBL8084982 0.86 KIF11 (0.38) IDO1TDO2ALDH1A1
SCHEMBL8097966 0.85 KIF11 (0.37) IDO1TDO2ALDH1A1PIK3CAMTOR
SCHEMBL8090834 0.85 KIF11 (0.35) IDO1TDO2ALDH1A1
SCHEMBL8091026 0.82 NAMPT (0.36) IDO1TDO2ALDH1A1PIK3CAMTOR
SCHEMBL8090786 0.82 SGK1 (0.37) SGK1ALDH1A1MTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007748-A2 TRISUBSTITUTED PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PROLIFERATIVE DISEASES ASTRAZENECA AB (SE) 2009-01-15 WO disclosed