SCHEMBL8083416

SCHEMBL8083416

NC(=O)Nc1ccc(-c2nc(N)cc(C3(S(=O)(=O)c4ccccc4F)CC3)n2)cc1

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PIK3R1 P27986 1/20 0.39
PIK3CA P42336 1/20 0.39
SGK1 O00141 11/20 0.38
ALOX5AP P20292 2/20 0.35
FEN1 P39748 2/20 0.35
IDO1 P14902 1/20 0.34
TDO2 P48775 1/20 0.34
F10 P00742 1/20 0.34
KIF11 P52732 1/20 0.34
MEN1 O00255 2/20 0.33
ALDH1A1 P00352 2/20 0.33
MAPT P10636 2/20 0.33
HPGD P15428 2/20 0.33
KMT2A Q03164 2/20 0.33
NAMPT P43490 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
KDM4E B2RXH2 1/20 0.33
CYP2C19 P33261 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8104712 0.90 IDO1 (0.40) PIK3CASGK1IDO1TDO2KIF11
SCHEMBL8082685 0.90 IDO1 (0.40) PIK3CASGK1IDO1TDO2ALDH1A1
SCHEMBL8090834 0.89 KIF11 (0.35) IDO1TDO2KIF11MEN1ALDH1A1
SCHEMBL8090786 0.89 SGK1 (0.37) SGK1F10MEN1ALDH1A1MAPT
SCHEMBL8091143 0.89 KIF11 (0.36) PIK3CASGK1F10KIF11MEN1
SCHEMBL8096684 0.87 NAMPT (0.39) PIK3R1PIK3CASGK1ALOX5APFEN1
SCHEMBL8095173 0.87 NAMPT (0.39) PIK3R1PIK3CASGK1MAPTNAMPT
SCHEMBL8091293 0.86 MAPT (0.42) PIK3R1PIK3CAKIF11MEN1ALDH1A1
SCHEMBL8091502 0.86 NAMPT (0.39) PIK3R1PIK3CASGK1MAPTNAMPT
SCHEMBL8084982 0.85 KIF11 (0.38) IDO1TDO2KIF11MEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007748-A2 TRISUBSTITUTED PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PROLIFERATIVE DISEASES ASTRAZENECA AB (SE) 2009-01-15 WO disclosed