SCHEMBL8112930

SCHEMBL8112930

CC(C)c1ccc(NC(=O)CN(c2cccc(C#N)c2)C(CC(=O)OC(C)(C)C)c2c[nH]cn2)cc1

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.35
MAPT P10636 2/20 0.35
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34
MCHR1 Q99705 5/20 0.33
PANK3 Q9H999 1/20 0.33
MAP2K2 P36507 1/20 0.33
CALCRL Q16602 1/20 0.33
HTT P42858 1/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
HPGD P15428 1/20 0.33
PSMB5 P28074 1/20 0.33
RORC P51449 1/20 0.32
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
LMNA P02545 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8104039 0.88 RAB9A (0.35) ALDH1A1MAPTNPC1RAB9AMCHR1
SCHEMBL8118826 0.86 MAPT (0.38) ALDH1A1MAPTNPC1RAB9AMCHR1
SCHEMBL8113212 0.85 MAPT (0.38) ALDH1A1MAPTNPC1RAB9AMCHR1
SCHEMBL8112413 0.84 NLRP3 (0.36) ALDH1A1MAPTNPC1RAB9AMCHR1
SCHEMBL8104245 0.84 RORC (0.38) ALDH1A1MAPTRAB9APANK3HTT
SCHEMBL8104404 0.79 PSMB5 (0.36) ALDH1A1MAPTMCHR1MAP2K2CALCRL
Hydrochloric Acid SCHEMBL8118543 0.79 F2 (0.37) NPC1RAB9ASMN1; SMN2HPGDKMT2A
SCHEMBL8113483 0.77 NPC1 (0.35) ALDH1A1MAPTNPC1RAB9AMCHR1
Hydrochloric Acid SCHEMBL8104643 0.76 ITGB3 (0.34) MAPTNPC1RAB9ASMN1; SMN2HPGD
SCHEMBL8113521 0.76 MAPT (0.42) ALDH1A1MAPTNPC1RAB9AMCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1020434-A1 3-AMIDINOANILINE DERIVATIVES, ACTIVATED BLOOD COAGULATION FACTOR X INHIBITORS, AND INTERMEDIATES FOR PRODUCING BOTH Kissei Pharmaceutical Co., Ltd. (JP) 2000-07-19 EP disclosed