SCHEMBL8130697

SCHEMBL8130697

Brc1ccc(Oc2cccs2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.43
LTA4H P09960 1/20 0.40
TDP1 Q9NUW8 2/20 0.38
LMNA P02545 1/20 0.37
SLC6A2 P23975 1/20 0.35
SLC6A4 P31645 1/20 0.35
SLC6A3 Q01959 1/20 0.35
CES2 O00748 1/20 0.35
CES1 P23141 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
POLB P06746 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
KCNA5 P22460 1/20 0.34
ALDH1A1 P00352 3/20 0.33
TSHR P16473 2/20 0.33
MAOA P21397 1/20 0.33
MAOB P27338 1/20 0.33
CYP2A6 P11509 1/20 0.33
APP P05067 1/20 0.33
BACE1 P56817 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8471918 0.89 MGMT (0.37) MAPTLTA4HTDP1CES2CES1
SCHEMBL16561451 0.87 CES2 (0.50) MAPTTDP1LMNACES2CES1
SCHEMBL141870 0.80 LTA4H (0.50) MAPTLTA4HTSHRMAOAMAOB
SCHEMBL2876554 0.79 APP (0.33) L3MBTL1ALDH1A1APPBACE1MGMT
SCHEMBL8124374 0.79 MAOA (0.43) MAPTLTA4HLMNASLC6A2SLC6A4
SCHEMBL9479303 0.79 GAA (0.47) MAPTTDP1LMNASLC6A2SLC6A4
SCHEMBL251357 0.77 MGMT (0.40) MAPTTDP1LMNACES2CES1
SCHEMBL7565860 0.75 MGMT (0.33) APPBACE1MGMT
SCHEMBL3965732 0.75 ALDH1A1 (0.49) MAPTLMNASMN1; SMN2POLBL3MBTL1
SCHEMBL8125571 0.75 IDO1 (0.44) LTA4HSMN1; SMN2POLBL3MBTL1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1028945-A1 SUBSTITUTED PYRIDINE COMPOUNDS AS ANTI-INFLAMMATORY AGENTS Amgen Inc. (US) 2000-08-23 EP disclosed
WO-1999024404-A1 SUBSTITUTED PYRIDINE COMPOUNDS AS ANTI-INFLAMMATORY AGENTS AMGEN INC. (US) 1999-05-20 WO disclosed