SCHEMBL8137883

SCHEMBL8137883

N#Cc1ccc2c(c1)C(OS(=O)(=O)C(F)(F)F)=CC(CF)(CF)O2

nearest known ligand 0.34

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.34
AKR1C3 P42330 1/20 0.33
PDE4A P27815 1/20 0.33
PDE4C Q08493 1/20 0.33
PDE4D Q08499 1/20 0.33
BACE1 P56817 1/20 0.33
TRPV4 Q9HBA0 1/20 0.32
P2RY6 Q15077 1/20 0.31
KCNE1 P15382 3/20 0.31
KCNQ1 P51787 3/20 0.31
PTGDR2 Q9Y5Y4 2/20 0.31
MEN1 O00255 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C19 P33261 1/20 0.31
KMT2A Q03164 1/20 0.31
KCND3 Q9UK17 1/20 0.31
HTR2A P28223 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7034282 0.83 PTGDR2 (0.31) PTGS2PTGDR2
SCHEMBL8135352 0.79 PDE4A (0.34) PTGS2PDE4APDE4CPDE4DPTGDR2
SCHEMBL8312376 0.74 PTGS2 (0.38) PTGS2KCNE1KCNQ1PTGDR2MEN1
SCHEMBL8312895 0.69 GABRA1 (0.37) PTGS2KCNE1KCNQ1
SCHEMBL8314385 0.68 ABCC9 (0.36) KCNE1KCNQ1
SCHEMBL8133760 0.68 HTR1A (0.33) PDE4APDE4CPDE4DHTR2A
SCHEMBL16381648 0.67 KDM4E (0.40) PTGS2
SCHEMBL14666733 0.67 ALDH1A1 (0.35)
SCHEMBL6590616 0.66 CYP3A4 (0.35) P2RY6CYP3A4KMT2A
SCHEMBL2682796 0.66 HIF1A (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0655448-B1 BENZOPYRAN AND BENZOXAZINE DERIVATIVES CHUGAI PHARMACEUTICAL CO LTD (JP) 2000-04-12 EP disclosed
US-5977167-A Benzopyran and benzoxazine derivatives CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 1999-11-02 US disclosed
US-5874446-A ANTIASTHMATICS, ANTIEPILEPSY AGENTS CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 1999-02-23 US disclosed
US-5614633-A POTASSIUM CHANNEL ACTIVATOR CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 1997-03-25 US disclosed
EP-0655448-A1 BENZOPYRAN AND BENZOXAZINE DERIVATIVES CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 1995-05-31 EP disclosed