SCHEMBL8312376

SCHEMBL8312376

N#Cc1ccc2c(c1)C(C(=O)O)=CC(CF)(CF)O2

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.38
HTR2A P28223 1/20 0.35
PTGDR2 Q9Y5Y4 2/20 0.34
KDM4C Q9H3R0 1/20 0.34
ABCB1 P08183 5/20 0.33
KDM4E B2RXH2 1/20 0.33
XDH P47989 4/20 0.33
SLC22A12 Q96S37 4/20 0.33
ABCC9 O60706 1/20 0.32
CYP2C8 P10632 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP3A4 P08684 2/20 0.32
ALOX15 P16050 1/20 0.32
KCNE1 P15382 3/20 0.32
KCNQ1 P51787 3/20 0.32
MEN1 O00255 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C19 P33261 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8314385 0.85 ABCC9 (0.36) ABCB1KDM4EABCC9KCNE1KCNQ1
SCHEMBL8312895 0.83 GABRA1 (0.37) PTGS2ABCC9CYP2C9KCNE1KCNQ1
SCHEMBL8316738 0.82 ABCC9 (0.32) ABCC9
SCHEMBL8316452 0.76 OPRD1 (0.35) KDM4ECYP2C9MEN1CYP1A2CYP2C19
SCHEMBL8137883 0.74 PTGS2 (0.34) PTGS2HTR2APTGDR2CYP3A4KCNE1
SCHEMBL8133760 0.71 HTR1A (0.33) HTR2AABCC9
SCHEMBL8130466 0.70 ABCC9 (0.41) HTR2AKDM4EABCC9CYP2C9CYP1A2
SCHEMBL8123176 0.70 GRM5 (0.39) KDM4EMEN1KMT2A
SCHEMBL8131499 0.69 HTR2A (0.47) HTR2AKDM4ECYP3A4KCNE1KCNQ1
SCHEMBL8897866 0.69 PTGS1 (0.37) PTGS2PTGDR2KDM4EXDHSLC22A12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0632033-B1 NOVEL BENZOPYRAN DERIVATIVE CHUGAI PHARMACEUTICAL CO LTD (JP) 1999-04-07 EP disclosed
US-5646308-A POTASSIUM CHANNEL ACTIVATORS USED AS ANTIASTHMATICS, ANTIEPILEPTICS CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 1997-07-08 US disclosed
EP-0632033-A1 NOVEL BENZOPYRAN DERIVATIVE CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 1995-01-04 EP disclosed