SCHEMBL8153003

SCHEMBL8153003

CS(=O)(=O)c1ccc(-c2cccc(C(Cc3ncco3)C(=O)O)c2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSK P43235 3/20 0.48
CTSS P25774 2/20 0.48
PPARG P37231 2/20 0.40
PPARA Q07869 2/20 0.40
SYK P43405 1/20 0.39
PTGS2 P35354 2/20 0.39
LRRK2 Q5S007 1/20 0.38
CTSL P07711 1/20 0.37
CTSB P07858 1/20 0.37
CYP2C9 P11712 4/20 0.37
PDE4A P27815 3/20 0.37
PDE4B Q07343 3/20 0.37
PDE4C Q08493 3/20 0.37
PDE4D Q08499 3/20 0.37
CTSA P10619 3/20 0.37
KDM5A P29375 1/20 0.36
KDM4C Q9H3R0 1/20 0.36
KDM5B Q9UGL1 1/20 0.36
PSEN1 P49768 1/20 0.36
PSEN2 P49810 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8146329 0.90 CTSK (0.47) CTSKCTSSPPARGPPARASYK
SCHEMBL5732085 0.90 CA2 (0.43) CTSKCTSSPPARGPPARASYK
SCHEMBL5732592 0.89 LNPEP (0.38) CTSKCTSSPPARGPPARACTSL
SCHEMBL5733048 0.80 CA2 (0.41) CTSKCTSSSYK
SCHEMBL5732778 0.78 LNPEP (0.37) CTSKCTSSCTSLCTSBKDM5A
SCHEMBL5732942 0.78 CA2 (0.43) CTSKCTSSCTSLCTSB
SCHEMBL5732590 0.69 PTGS2 (0.44) PTGS2CTSA
SCHEMBL8551224 0.69 CA2 (0.46) SYKLRRK2CTSA
SCHEMBL6581771 0.69 CTSS (0.51) CTSKCTSSPTGS2
SCHEMBL4714948 0.68 CTSK (0.57) CTSKCTSSCTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6090834-A ANALGESICS; RHEUMATIC DISORDERS; SKIN DISORDERS; GASTROINTESTINAL DISORDERS G.D. SEARLE & CO. (US) 2000-07-18 US disclosed
EP-0825989-A1 SUBSTITUTED OXAZOLES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1998-03-04 EP disclosed
WO-1996036617-A1 SUBSTITUTED OXAZOLES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-11-21 WO disclosed