Fumaric Acid

Fumaric Acid

SCHEMBL8162

CC(N)C#N.O=C(O)C=CC(=O)O

nearest known ligand 0.52

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Known targets — ChEMBL curated mechanism

ACEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ATP4AATP4BAXLBTKCACNA1CCACNA1DCACNA1FCACNA1SCCR5CHRM2CHRM3CPT1BCPT2DPP4DRD1DRD2EGFRERBB2ERBB4FLT3HRH1HRH3HTR1AHTR2AHTR2BHTR2CHTR4JAK1JAK2JAK3KCNH2KMT2AMAP2K1MAP2K2MEN1MLNRMPLMTORPPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PLK4PPARGRENS1PR1SLC6A2SLC6A3SLC6A4SMOTYK2atpAatpBatpCatpDatpEatpFatpFHatpGpol

The experimentally established mechanism targets of Fumaric Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 known ✓ O00255 1/20 0.46
KMT2A known ✓ Q03164 1/20 0.46
DPP4 known ✓ P27487 2/20 0.35
GABRP O00591 2/20 0.52
GABRD O14764 2/20 0.52
GABRA1 P14867 2/20 0.52
GABRB1 P18505 2/20 0.52
GABRG2 P18507 2/20 0.52
GABRB3 P28472 2/20 0.52
GABRA5 P31644 2/20 0.52
GABRA3 P34903 2/20 0.52
GABRA2 P47869 2/20 0.52
GABRB2 P47870 2/20 0.52
GABRA4 P48169 2/20 0.52
GABRE P78334 2/20 0.52
GABRA6 Q16445 2/20 0.52
GABRG1 Q8N1C3 2/20 0.52
GABRG3 Q99928 2/20 0.52
GABRQ Q9UN88 2/20 0.52
TSHR P16473 4/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fumaric Acid SCHEMBL138088 1.00 GABRP (0.52) GABRPGABRDGABRA1GABRB1GABRG2
Bicarbonate SCHEMBL4001353 0.84
Maleic Acid SCHEMBL8957408 0.81 GABRP (0.65) GABRPGABRDGABRA1GABRB1GABRG2
Fumaric Acid SCHEMBL21145282 0.81 GABRP (0.65) GABRPGABRDGABRA1GABRB1GABRG2
Fumaric Acid SCHEMBL21145284 0.81 GABRP (0.65) GABRPGABRDGABRA1GABRB1GABRG2
Maleic Acid SCHEMBL3118041 0.78 GABRP (0.62) GABRPGABRDGABRA1GABRB1GABRG2
Fumaric Acid SCHEMBL1835364 0.78 GABRP (0.62) GABRPGABRDGABRA1GABRB1GABRG2
Fumaric Acid SCHEMBL1835366 0.78 GABRP (0.62) GABRPGABRDGABRA1GABRB1GABRG2
Formic Acid SCHEMBL20504179 0.76
Formic Acid SCHEMBL20504180 0.76

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2760 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025133663-A1 DIGITAL TISSUE REPAIR MODEL Institut National de la Santé et de la Recherche Médicale (FR) 2025-06-26 WO claimed
CN-119074707-A Research and application of alkaloid compound in prevention and treatment of abdominal aortic aneurysm 上海市第十人民医院 2024-12-06 CN claimed
CN-117045628-A Research and application of alkaloid compound in prevention and treatment of abdominal aortic aneurysm 上海市第十人民医院 2023-11-14 CN claimed
US-8114152-B2 Stent coating ICON INTERVENTIONAL SYSTEMS, INC. (US) 2012-02-14 US claimed
US-20090062904-A1 STENT COATING ICON INTERVENTIONAL SYSTEMS, INC. 2009-03-05 US claimed
EP-1738759-A1 Inhibition of abnormal cell proliferation with camptothecin and combinations including the same SuperGen, Inc. (US) 2007-01-03 EP claimed
US-20050118180-A1 Inhibition of abnormal cell proliferation with camptothecin and combinations including the same SUPERGEN, INC. 2005-06-02 US claimed
EP-1276479-A2 INHIBITION OF ABNORMAL CELL PROLIFERATION WITH CAMPTOTHECIN AND COMBINATIONS INCLUDING THE SAME SuperGen, Inc. (US) 2003-01-22 EP claimed
US-20020111362-A1 Inhibition of abnormal cell proliferation with camptothecin and combinations including the same SUPERGEN, INC. 2002-08-15 US claimed
WO-2001080843-A2 INHIBITION OF ABNORMAL CELL PROLIFERATION WITH CAMPTOTHECIN AND COMBINATIONS INCLUDING THE SAME SUPERGEN, INC. (US) 2001-11-01 WO claimed
EP-0564722-A1 Lathyrogenic agents and apparatus for the treatment of fibrotic lesions LATHROTEC INC (US) 1993-10-13 EP claimed
US-5120322-A Method and apparatus for treatment of fibrotic lesions LATHROTEC, INC. (US) 1992-06-09 US claimed
EP-3325513-B1 ANTI-PD-L1 ANTIBODIES AND USES THEREOF I MAB BIOPHARMA CO LTD (CN) 2026-05-20 EP disclosed
US-20260130893-A1 PRMT5 INHIBITORS AND USES THEREOF GILEAD SCIENCES INC (US) 2026-05-14 US disclosed
EP-4735445-A1 KRAS MODULATING COMPOUNDS GILEAD SCIENCES, INC. (US) 2026-05-06 EP disclosed
EP-4735453-A1 KRAS MODULATING COMPOUNDS GILEAD SCIENCES, INC. (US) 2026-05-06 EP disclosed
US-4820843-A Tetrazole intermediates to antihypertensive compounds E. I. DU PONT DE NEMOURS AND COMPANY (US) 1989-04-11 US disclosed
EP-0291969-A2 Tetrazole intermediates to antihypertensive compounds E.I. DU PONT DE NEMOURS AND COMPANY (US) 1988-11-23 EP disclosed
US-4485088-A INHIBITION OF ABNORMAL SCAR FORMATION BIO-PRODUCTS, INC. (US) 1984-11-27 US disclosed
US-4485088-A INHIBITION OF ABNORMAL SCAR FORMATION BIO-PRODUCTS, INC. (US) 1984-11-27 US disclosed