SCHEMBL816348

SCHEMBL816348

Cc1ccc(N(C(F)(F)F)C(F)(F)F)cc1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.48
TSHR P16473 2/20 0.48
ACHE P22303 5/20 0.42
TDP1 Q9NUW8 1/20 0.42
CA2 P00918 3/20 0.35
MAPT P10636 2/20 0.35
CA1 P00915 2/20 0.35
CA9 Q16790 2/20 0.35
MCOLN3 Q8TDD5 1/20 0.35
CYP2C19 P33261 1/20 0.35
CA5A P35218 1/20 0.35
CA7 P43166 1/20 0.33
MLYCD O95822 1/20 0.32
CHRNA7 P36544 1/20 0.32
RORC P51449 1/20 0.32
NFE2L2 Q16236 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12828075 0.77 ALDH1A1 (0.52) ALDH1A1TSHRACHETDP1CA2
SCHEMBL3615102 0.74 ALDH1A1 (0.46) ALDH1A1TSHRACHETDP1MAPT
SCHEMBL12749948 0.73 PTPN5 (0.38) ALDH1A1
SCHEMBL728216 0.72 ALDH1A1 (0.41) ALDH1A1TSHRTDP1CA2MAPT
SCHEMBL132308 0.72 ALDH1A1 (0.46) ALDH1A1TSHRACHETDP1CA2
SCHEMBL2137923 0.72 ALDH1A1 (0.46) ALDH1A1TSHRACHETDP1CA2
SCHEMBL816352 0.72 ACHE (0.46) ALDH1A1ACHETDP1MAPTCYP2C19
SCHEMBL9999807 0.69 TSHR (0.42) ALDH1A1TSHRACHECA2CA1
SCHEMBL19356905 0.68
SCHEMBL16982395 0.67 ALDH1A1 (0.61) ALDH1A1TSHRACHETDP1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1805158-B1 SULFONYL-SUBSTITUTED BICYCLIC COMPOUNDS AS MODULATORS OF PPAR KALYPSYS INC (US) 2018-06-27 EP disclosed
US-8067625-B2 Fluorosurfactants MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2011-11-29 US disclosed
US-8049022-B2 Fluorosurfactants MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2011-11-01 US disclosed
US-7834004-B2 Sulfonyl-substituted bicyclic compounds as modulators of PPAR KALYPSYS, INC (US) 2010-11-16 US disclosed
US-20100152081-A1 Fluorosurfactants MERCK PATENT GMBH (DE) 2010-06-17 US disclosed
US-20090312432-A1 FLUOROSURFACTANTS MERCK PATENT GESELLSCHAFT (DE) 2009-12-17 US disclosed
US-20090264525-A1 FLUOROSURFACTANTS MERCK PATENT GMBH (DE) 2009-10-22 US disclosed
US-20090264417-A1 SULFONYL-SUBSTITUTED BICYCLIC COMPOUNDS AS MODULATORS OF PPAR KALYPSYS, INC. (US) 2009-10-22 US disclosed
US-20090227599-A1 SULFONYL-SUBSTITUTED BICYCLIC COMPOUNDS AS MODULATORS OF PPAR KALYPSYS, INC. (US) 2009-09-10 US disclosed
US-7517884-B2 {5-[4-(4-Trifluoromethyl-phenyl)-piperazine-1-sulfonyl]-indan-2-yl}-acetic acid; peroxisome proliferator activated receptors modulator; antidiabetic, antiinflammatory agent; obesity, hyperinsulinemia, metabolic syndrome X, polycystic ovary syndrome, ischemia-associated organ injury, diabetes KALYPSYS INC. (US) 2009-04-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090312432-A1 FLUOROSURFACTANTS SGMS2, FASN, SGMS1 ALDH1A1 2479/4885TSHR 1160/4885ACHE 4091/4885
US-20100152081-A1 Fluorosurfactants CBR3, FPR3, NOX3 ALDH1A1 2466/4885TSHR 886/4885ACHE 3673/4885
US-20090227599-A1 SULFONYL-SUBSTITUTED BICYCLIC COMPOUNDS AS MODULATORS OF PPAR PPARG, PPARA, PPARD ALDH1A1 1551/4885TSHR 262/4885ACHE 2442/4885
US-20090264525-A1 FLUOROSURFACTANTS FASN, FFAR3, SGMS2 ALDH1A1 2925/4885TSHR 754/4885ACHE 4537/4885
US-20090264417-A1 SULFONYL-SUBSTITUTED BICYCLIC COMPOUNDS AS MODULATORS OF PPAR PPARG, PPARA, PPARD ALDH1A1 1551/4885TSHR 262/4885ACHE 2442/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.