SCHEMBL8167287

SCHEMBL8167287

CCN(Cc1cc(Br)ccc1OCc1occc1C)c1ccc(C(=O)O)cn1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HCAR3 P49019 2/20 0.41
RXRA P19793 9/20 0.37
PTGER1 P34995 6/20 0.37
RXRB P28702 1/20 0.36
RXRG P48443 1/20 0.36
GBA1 P04062 1/20 0.36
KDM5A P29375 1/20 0.35
KDM4C Q9H3R0 1/20 0.35
KDM5B Q9UGL1 1/20 0.35
CYP1A2 P05177 1/20 0.35
PPARG P37231 1/20 0.35
CCR5 P51681 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8168017 0.91 MEN1 (0.35) HCAR3PTGER1GBA1CYP1A2CCR5
SCHEMBL8703967 0.84 CCR5 (0.48) HCAR3RXRAPTGER1RXRBCYP1A2
SCHEMBL8701112 0.83 CCR5 (0.46) HCAR3RXRAPTGER1CYP1A2CCR5
SCHEMBL1907786 0.83 RXRA (0.53) HCAR3RXRAPTGER1CYP1A2CCR5
SCHEMBL7672615 0.82 HCAR3 (0.51) HCAR3RXRAGBA1PPARG
SCHEMBL8162210 0.81 ALDH1A1 (0.45) HCAR3RXRAPTGER1CYP1A2CCR5
SCHEMBL8167622 0.81 GAA (0.48) HCAR3RXRAPTGER1GBA1CYP1A2
SCHEMBL8167606 0.81 CCR5 (0.58) RXRAPTGER1CCR5
SCHEMBL7673319 0.80 RXRA (0.56) HCAR3RXRAPTGER1RXRBRXRG
SCHEMBL7974626 0.79 HCAR3 (0.46) HCAR3RXRAGBA1PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0773930-B1 AROMATIC AMINO ETHERS AS PAIN RELIEVING AGENTS ZENECA LTD (GB) 2000-10-11 EP disclosed
US-5843942-A Aromatic amino ethers as pain relieving agents ZENECA LIMITED (GB) 1998-12-01 US disclosed