SCHEMBL8169641

SCHEMBL8169641

CC(C)(C)NS(=O)(=O)c1ccc(C(=N)N)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TMPRSS6 Q8IU80 3/20 0.55
ALDH1A1 P00352 5/20 0.51
MAPT P10636 2/20 0.51
SMN1; SMN2 Q16637 2/20 0.51
F2 P00734 2/20 0.49
PRSS1 P07477 2/20 0.49
PRSS2 P07478 2/20 0.49
PRSS3 P35030 2/20 0.49
CYP3A4 P08684 1/20 0.47
CYP2C9 P11712 1/20 0.47
MAPK1 P28482 1/20 0.47
HPN P05981 3/20 0.45
PLAU P00749 2/20 0.45
LMNA P02545 2/20 0.45
HPGD P15428 2/20 0.45
KDM4E B2RXH2 1/20 0.45
MEN1 O00255 1/20 0.45
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
KMT2A Q03164 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5458574 0.84 CA2 (0.53) ALDH1A1MAPTSMN1; SMN2CYP3A4CYP2C9
SCHEMBL14448891 0.80 TMPRSS6 (0.60) TMPRSS6ALDH1A1SMN1; SMN2F2PRSS1
SCHEMBL3716571 0.79 ALDH1A1 (0.54) ALDH1A1MAPTSMN1; SMN2F2PRSS1
SCHEMBL3643243 0.79 ALDH1A1 (0.58) ALDH1A1MAPTSMN1; SMN2CYP3A4CYP2C9
SCHEMBL2408403 0.76 ALDH1A1 (0.59) ALDH1A1MAPTSMN1; SMN2CYP3A4CYP2C9
SCHEMBL1479992 0.76 ALDH1A1 (0.59) ALDH1A1MAPTSMN1; SMN2CYP3A4CYP2C9
SCHEMBL12348122 0.75 TMPRSS6 (0.58) TMPRSS6ALDH1A1F2PRSS1PRSS2
SCHEMBL8486571 0.75 ALDH1A1 (0.64) ALDH1A1MAPTSMN1; SMN2CYP3A4CYP2C9
SCHEMBL7895365 0.75 MEN1 (0.54) ALDH1A1MAPTSMN1; SMN2CYP3A4CYP2C9
SCHEMBL8724306 0.75 ALDH1A1 (0.50) ALDH1A1MAPTSMN1; SMN2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250162989-A1 USP30 INHIBITORS AND USES THEREOF VINCERE BIOSCIENCES, INC. 2025-05-22 US disclosed
CN-117836270-A USP30 inhibitors and uses thereof 文森雷生物科学股份有限公司 2024-04-05 CN disclosed
EP-4305021-A1 USP30 INHIBITORS AND USES THEREOF Vincere Biosciences, Inc. (US) 2024-01-17 EP disclosed
WO-2022192562-A1 USP30 INHIBITORS AND USES THEREOF VINCERE BIOSCIENCES, INC. (US) 2022-09-15 WO disclosed
US-6114328-A ANTICOAGULANTS; BLOOD DISORDERS DUPONT PHARMACEUTICALS COMPANY (US) 2000-09-05 US disclosed
US-5849736-A Isoxazoline and isoxazole fibrinogen receptor antagonists THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1998-12-15 US disclosed
EP-0730590-A1 NOVEL ISOXAZOLINE AND ISOXAZOLE FIBRINOGEN RECEPTOR ANTAGONISTS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-09-11 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250162989-A1 USP30 INHIBITORS AND USES THEREOF USP30, USP28, USP1 TMPRSS6 2305/4885ALDH1A1 2021/4885MAPT 2434/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.