SCHEMBL8199744

SCHEMBL8199744

C=C(C)c1ccc(-c2c(Cl)n[nH]c2-c2ccc([S+](C)[O-])cc2)cc1

nearest known ligand 0.35

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
RPS6KA3 P51812 1/20 0.32
MAPK1 P28482 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
MAPK13 O15264 1/20 0.30
MAPK12 P53778 1/20 0.30
MAPK11 Q15759 1/20 0.30
MAPK14 Q16539 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8200029 0.88 XDH (0.39) RPS6KA3MAPK1NPSR1MAPK13MAPK12
SCHEMBL8637992 0.82 MAPK14 (0.46) RPS6KA3MAPK1NPSR1MAPK13MAPK12
SCHEMBL8194840 0.78 MAPT (0.37) MAPK1NPSR1MAPK14
SCHEMBL8196956 0.75 CA2 (0.36)
SCHEMBL8199102 0.73 ALDH1A1 (0.36)
SCHEMBL8196073 0.67 ENPP1 (0.35) RPS6KA3MAPK1NPSR1MAPK14
SCHEMBL8201330 0.66 SMN1; SMN2 (0.39)
SCHEMBL8640165 0.66 RPS6KA3 (0.33) RPS6KA3MAPK1NPSR1
SCHEMBL8201683 0.64 MAPK14 (0.44) RPS6KA3MAPK1NPSR1MAPK13MAPK12
SCHEMBL8195581 0.63 LMNA (0.39) RPS6KA3MAPK1NPSR1MAPK13MAPK12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000018741-A2 PYRAZOLE COMPOUNDS AS COX-2 INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-04-06 WO disclosed