SCHEMBL8199872

SCHEMBL8199872

CC(C)c1cc(C(=O)NC(Cc2ccccc2)C2=COCO2)c(N)s1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.44
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
KMT2A Q03164 2/20 0.35
MEN1 O00255 1/20 0.35
GAA P10253 3/20 0.34
MAPT P10636 2/20 0.34
GFER P55789 1/20 0.34
ALDH1A1 P00352 3/20 0.34
ALOX15 P16050 2/20 0.34
TACR3 P29371 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HTT P42858 1/20 0.33
GLA P06280 2/20 0.33
MCL1 Q07820 1/20 0.33
HPGD P15428 1/20 0.33
ABCC2 Q92887 1/20 0.33
GALR1 P47211 1/20 0.33
PSMB5 P28074 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8209525 0.88 KMT2A (0.37) NPC1RAB9AKMT2AMEN1GAA
SCHEMBL8207229 0.87 ALOX15 (0.40) KMT2AGAAMAPTGFERALDH1A1
SCHEMBL8211806 0.86 PYGL (0.36) KMT2AMEN1GAAMAPTGFER
SCHEMBL8212891 0.86 ALDH1A1 (0.40) KMT2AMEN1GAAMAPTGFER
SCHEMBL8200315 0.85 ALOX15 (0.40) KMT2AALDH1A1ALOX15SMN1; SMN2HPGD
SCHEMBL8200038 0.84 NPC1 (0.37) NPC1RAB9AKMT2AMEN1MAPT
SCHEMBL8198895 0.82 SMN1; SMN2 (0.38) NPC1RAB9AKMT2AMEN1GAA
SCHEMBL8206432 0.74 TAAR1 (0.54) TAAR1NPC1RAB9AKMT2AMEN1
SCHEMBL8212479 0.74 MAPT (0.38) NPC1RAB9AKMT2AMEN1GAA
SCHEMBL8207755 0.73 GRIN2C (0.48) NPC1RAB9AKMT2AMEN1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6143777-A ENZYME INHIBITORS MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-11-07 US disclosed