SCHEMBL8200315

SCHEMBL8200315

CCCCc1cc(C(=O)NC(Cc2ccccc2)C2=COCO2)c(N)s1

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 5/20 0.40
GALR1 P47211 1/20 0.37
CNR1 P21554 3/20 0.36
CNR2 P34972 3/20 0.36
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HPGD P15428 1/20 0.35
CCNE1 P24864 1/20 0.34
CDK2 P24941 1/20 0.34
CDK5 Q00535 1/20 0.34
TP53 P04637 1/20 0.34
KMT2A Q03164 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8212891 0.95 ALDH1A1 (0.40) ALOX15GALR1CNR1CNR2KDM4E
SCHEMBL8207229 0.92 ALOX15 (0.40) ALOX15GALR1CNR1CNR2ALDH1A1
SCHEMBL8209525 0.87 KMT2A (0.37) ALOX15ALDH1A1KMT2ASMN1; SMN2
SCHEMBL8199872 0.85 TAAR1 (0.44) ALOX15GALR1ALDH1A1HPGDKMT2A
SCHEMBL8211806 0.85 PYGL (0.36) ALDH1A1HPGDKMT2ASMN1; SMN2
SCHEMBL8206045 0.84 GRIN2C (0.39) GALR1KDM4EALDH1A1HPGDKMT2A
SCHEMBL8199938 0.82 ALDH1A1 (0.38) GALR1KDM4EALDH1A1HPGDKMT2A
SCHEMBL8206226 0.80 ALDH1A1 (0.42) ALOX15KDM4EALDH1A1HPGDKMT2A
SCHEMBL8200375 0.78 ALDH1A1 (0.41) ALOX15CNR1CNR2KDM4EALDH1A1
SCHEMBL8207755 0.76 GRIN2C (0.48) KDM4EALDH1A1HPGDKMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6143777-A ENZYME INHIBITORS MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-11-07 US disclosed