SCHEMBL8200595

SCHEMBL8200595

COc1ccc(OC)c(NC(=O)c2cccc3c2CCC(CCN2CCC(c4ccccc4)CC2)C3=O)c1

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.45
MAPT P10636 2/20 0.44
KDM4E B2RXH2 1/20 0.44
LMNA P02545 1/20 0.44
HPGD P15428 1/20 0.44
TSHR P16473 1/20 0.44
ATM Q13315 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
HSD17B10 Q99714 1/20 0.44
GFER P55789 1/20 0.44
CCR5 P51681 4/20 0.44
POLB P06746 2/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.43
HTR2C P28335 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8203549 0.87 HTR2C (0.43) ALDH1A1KDM4ETSHRNPSR1MEN1
SCHEMBL8200188 0.84 KDM4E (0.44) KDM4EMEN1KMT2ASMN1; SMN2HTR2C
SCHEMBL8200414 0.83 PRCP (0.44) ALDH1A1ATMCCR5MEN1KMT2A
SCHEMBL8199643 0.81 CCR5 (0.48) CCR5HTR2C
SCHEMBL8200402 0.78 HTR2C (0.48) CCR5HTR2C
SCHEMBL8199345 0.78 CCR2 (0.46) CCR5HTR2C
SCHEMBL8191618 0.78 HTR2C (0.50) ALDH1A1MAPTKDM4ECCR5POLB
SCHEMBL8198484 0.77 HTR2C (0.42) TSHRMEN1KMT2AHTR2C
SCHEMBL8192538 0.77 PRCP (0.56) ALDH1A1KDM4ELMNAHPGDHSD17B10
SCHEMBL8199832 0.77 PRCP (0.56) ALDH1A1KDM4ELMNAHPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6048877-A Tetralone derivatives as antiarrhythmic agents BRISTOL-MYERS SQUIBB COMPANY (US) 2000-04-11 US claimed
WO-1998036749-A1 TETRALONE DERIVATIVES AS ANTIARRHYTHMIC AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 1998-08-27 WO claimed
US-6048877-A Tetralone derivatives as antiarrhythmic agents BRISTOL-MYERS SQUIBB COMPANY (US) 2000-04-11 US disclosed