SCHEMBL8208503

SCHEMBL8208503

CONC(=O)c1cc(Cl)ccc1N

nearest known ligand 0.58

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
FADS1 O60427 2/20 0.56
ABL1 P00519 1/20 0.56
GCK P35557 2/20 0.51
RECQL P46063 1/20 0.50
NOS2 P35228 2/20 0.47
ALDH1A1 P00352 4/20 0.46
LMNA P02545 1/20 0.45
KDM4E B2RXH2 2/20 0.44
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
BRAF P15056 1/20 0.44
HDAC1 Q13547 1/20 0.44
GLA P06280 1/20 0.44
GAA P10253 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8205593 0.86 ABL1 (0.70) FADS1ABL1ALDH1A1LMNAKDM4E
SCHEMBL140037 0.82 FADS1 (0.59) FADS1ABL1GCKRECQLNOS2
SCHEMBL267531 0.82 ABL1 (0.74) FADS1ABL1RECQLNOS2ALDH1A1
SCHEMBL13761455 0.81 FADS1 (0.55) FADS1ABL1GCKRECQLNOS2
SCHEMBL8639956 0.81 ALDH1A1 (0.66) ABL1RECQLALDH1A1LMNAKDM4E
SCHEMBL3637360 0.80 FADS1 (0.61) FADS1ABL1GCKRECQLNOS2
SCHEMBL1095186 0.80 ALDH1A1 (0.70) FADS1ABL1GCKRECQLNOS2
SCHEMBL28903979 0.80 LMNA (0.50) ABL1RECQLALDH1A1LMNAKDM4E
SCHEMBL15284054 0.79 KDM4E (0.58) RECQLALDH1A1KDM4ENPC1HDAC1
SCHEMBL8199077 0.79 BRAF (0.51) RECQLNOS2ALDH1A1KDM4ENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0979227-A1 4,1-BENZOXAZEPINES, THEIR ANALOGUES, AND THEIR USE AS SOMATOSTATIN AGONISTS Takeda Chemical Industries, Ltd. (JP) 2000-02-16 EP disclosed
WO-1998047882-A1 4,1-BENZOXAZEPINES, THEIR ANALOGUES, AND THEIR USE AS SOMATOSTATIN AGONISTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-10-29 WO disclosed