SCHEMBL8258997

SCHEMBL8258997

Fc1cc(Cl)c(-c2cccc3c2OCCC3)c(Cl)c1

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 6/20 0.38
CDK2 P24941 2/20 0.36
CDK9 P50750 2/20 0.36
HTR7 P34969 2/20 0.36
AQP1 P29972 1/20 0.35
PDK2 Q15119 1/20 0.33
GRM2 Q14416 2/20 0.33
NOTUM Q6P988 1/20 0.32
PARP1 P09874 1/20 0.32
MEN1 O00255 1/20 0.32
GAA P10253 1/20 0.32
CASP6 P55212 1/20 0.32
KMT2A Q03164 1/20 0.32
P2RX7 Q99572 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8256849 0.90 PARP1 (0.34) HTR1ACDK2CDK9HTR7NOTUM
SCHEMBL8259987 0.85 HTR1A (0.35) HTR1ACDK2CDK9HTR7
SCHEMBL8248843 0.83 LMNA (0.36) HTR1ACDK2CDK9PARP1GAA
SCHEMBL8259066 0.82 ALDH1A1 (0.36) HTR7GAAKMT2A
SCHEMBL8258142 0.82 XDH (0.35) CDK2CDK9NOTUMPARP1
SCHEMBL8256879 0.79 AQP1 (0.47) HTR1AAQP1NOTUMPARP1
SCHEMBL8254801 0.78 HTR1A (0.36) HTR1ACDK2CDK9AQP1NOTUM
SCHEMBL15319473 0.74 PARP1 (0.41) HTR1ANOTUMPARP1
SCHEMBL30543420 0.74 PARP1 (0.41) HTR1ANOTUMPARP1
SCHEMBL8248841 0.73 XDH (0.34) HTR1AAQP1NOTUMPARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006116165-A1 CHROMANE AND CHROMENE DERIVATIVES AND USES THEREOF WYETH (US) 2006-11-02 WO disclosed