SCHEMBL8259062

SCHEMBL8259062

Fc1ccc2[nH]cc(I)c2c1

nearest known ligand 0.58

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GPR84 Q9NQS5 2/20 0.58
MPO P05164 11/20 0.55
HTR2A P28223 3/20 0.51
TRPM8 Q7Z2W7 1/20 0.51
HTR1A P08908 1/20 0.50
KMT2A Q03164 1/20 0.50
HTR2C P28335 2/20 0.49
TSHR P16473 1/20 0.49
KDM4E B2RXH2 1/20 0.49
HTR2B P41595 1/20 0.49
SLC6A4 P31645 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2112913 0.83 GPR84 (0.58) GPR84HTR2A
SCHEMBL25045531 0.78 SLC6A4 (0.47) GPR84HTR2AHTR1ASLC6A4
SCHEMBL20584073 0.78 GPR84 (0.62) GPR84MPOHTR2ATRPM8HTR1A
SCHEMBL9268634 0.76 NR4A2 (0.68) GPR84MPOHTR2ATRPM8HTR1A
SCHEMBL16697905 0.76 GPR84 (0.57) GPR84MPOHTR2ATRPM8HTR1A
SCHEMBL208748 0.75 GPR84 (0.58) GPR84MPOHTR2ATRPM8HTR1A
SCHEMBL14631802 0.75 GPR84 (0.58) GPR84MPOHTR2ATRPM8HTR1A
SCHEMBL1372357 0.75 GPR84 (0.58) GPR84MPOHTR2ATRPM8HTR1A
SCHEMBL15623086 0.75 GPR84 (0.58) GPR84MPOHTR2ATRPM8HTR1A
SCHEMBL3624363 0.75 MPO (0.59) GPR84MPOHTR2ATRPM8HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 29 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12570632-B2 Indole derivatives and uses thereof for treating a cancer UNIVERSITE CLAUDE BERNARD LYON 1 (FR) 2026-03-10 US disclosed
EP-4175718-B1 INDOLE DERIVATIVES AND USES THEREOF FOR TREATING A CANCER UNIV CLAUDE BERNARD LYON (FR) 2024-10-02 EP disclosed
CN-115843271-B Indole derivatives and their use for the treatment of cancer 克洛德贝纳尔-里昂第一大学 2024-08-13 CN disclosed
EP-3583644-B1 ELECTRODE MATERIALS AND PROCESSES FOR THEIR PREPARATION HYDRO QUEBEC (CA) 2024-08-07 EP disclosed
EP-4090660-B1 QUINOXALINE DERIVATIVES GRUENENTHAL GMBH (DE) 2024-01-31 EP disclosed
US-20230278983-A1 INDOLE DERIVATIVES AND USES THEREOF FOR TREATING A CANCER UNIVERSITE CLAUDE BERNARD LYON 1 (FR) 2023-09-07 US disclosed
US-20230278983-A1 INDOLE DERIVATIVES AND USES THEREOF FOR TREATING A CANCER UNIVERSITE CLAUDE BERNARD LYON 1 (FR) 2023-09-07 US disclosed
EP-3805214-B1 JAK3 SELECTIVE INHIBITOR UNIV PEKING SHENZHEN GRADUATE SCHOOL (CN) 2023-07-05 EP disclosed
EP-4175718-A1 INDOLE DERIVATIVES AND USES THEREOF FOR TREATING A CANCER UNIVERSITE CLAUDE BERNARD - LYON 1 (FR) 2023-05-10 EP disclosed
CN-115843271-A Indole derivatives and their use for the treatment of cancer 克洛德贝纳尔-里昂第一大学 2023-03-24 CN disclosed
EP-3805214-A1 JAK3 SELECTIVE INHIBITOR Peking University Shenzhen Graduate School (CN) 2021-04-14 EP disclosed
US-20200052302-A1 ELECTRODE MATERIALS AND PROCESSES FOR THEIR PREPARATION HYDRO-QUéBEC (CA) 2020-02-13 US disclosed
US-20200052302-A1 ELECTRODE MATERIALS AND PROCESSES FOR THEIR PREPARATION HYDRO-QUéBEC (CA) 2020-02-13 US disclosed
US-20190263802-A1 COMPOUNDS AND METHOD OF USE MOLECULAR SKIN THERAPEUTICS, INC. 2019-08-29 US disclosed
WO-2018148833-A1 ELECTRODE MATERIALS AND PROCESSES FOR THEIR PREPARATION HYDRO-QUéBEC (CA) 2018-08-23 WO disclosed
EP-2961742-B1 AMIDE COMPOUNDS FOR THE TREATMENT OF HIV GILEAD SCIENCES INC (US) 2018-08-01 EP disclosed
EP-1827427-B1 ARYLOXYETHYLAMINE DERIVATIVES WITH A COMBINATION OF PARTIAL DOPAMINE-D2 RECEPTOR AGONISM AND SEROTONIN REUPTAKE INHIBITION SOLVAY PHARM BV (NL) 2008-07-23 EP disclosed
US-20070142397-A2 PHENYPIPERAZINE DERIVATIVES WITH A COMBINATION OF PARTIAL DOPAMINE-D2 RECEPTOR AGONISM AND SEROTONIN REUPTAKE INHIBITION SOLVAY PHARMECEUTICALS B.V. (NL) 2007-06-21 US disclosed
US-20070142397-A2 PHENYPIPERAZINE DERIVATIVES WITH A COMBINATION OF PARTIAL DOPAMINE-D2 RECEPTOR AGONISM AND SEROTONIN REUPTAKE INHIBITION SOLVAY PHARMECEUTICALS B.V. (NL) 2007-06-21 US disclosed
WO-2006061379-A1 PHENYLPIPERAZINE DERIVATIVES WITH A COMBINATION OF PARTIAL DOPAMINE-D2 RECEPTOR AGONISM AND SEROTONIN REUPTAKE INHIBITION SOLVAY PHARMACEUTICALS B.V. (NL) 2006-06-15 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200052302-A1 ELECTRODE MATERIALS AND PROCESSES FOR THEIR PREPARATION ALPL, EPCAM, MB GPR84 4720/4885MPO 85/4885HTR2A 4453/4885
US-12570632-B2 Indole derivatives and uses thereof for treating a cancer CKS2, CSNK2A3, CSNK1A1L GPR84 1655/4885MPO 4458/4885HTR2A 179/4885
US-20230278983-A1 INDOLE DERIVATIVES AND USES THEREOF FOR TREATING A CANCER CSNK2A1, IDO1, CSNK2A3 GPR84 1862/4885MPO 4538/4885HTR2A 293/4885
US-20190263802-A1 COMPOUNDS AND METHOD OF USE AIFM2, GPX4, GPX1 GPR84 2869/4885MPO 326/4885HTR2A 3059/4885
US-20070142397-A2 PHENYPIPERAZINE DERIVATIVES WITH A COMBINATION OF PARTIAL DOPAMINE-D2 RECEPTOR AGONISM AND SEROTONIN REUPTAKE INHIBITION HTR2C, HTR2A, HTR5A GPR84 203/4885MPO 4022/4885HTR2A 2/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.