SCHEMBL8288650

SCHEMBL8288650

Cc1sc(NC(=O)c2ccccc2F)c(C(N)=O)c1C

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 11/20 0.68
HPGD P15428 6/20 0.68
KDM4E B2RXH2 6/20 0.68
LMNA P02545 4/20 0.68
RAB9A P51151 7/20 0.60
NPC1 O15118 6/20 0.60
SMN1; SMN2 Q16637 6/20 0.60
TP53 P04637 2/20 0.60
MAPK10 P53779 1/20 0.60
HSD17B10 Q99714 1/20 0.60
MAPT P10636 11/20 0.59
MEN1 O00255 5/20 0.59
KMT2A Q03164 5/20 0.59
GAA P10253 3/20 0.59
MAPK1 P28482 2/20 0.56
NPSR1 Q6W5P4 2/20 0.56
NFKB1 P19838 1/20 0.56
CASP1 P29466 1/20 0.56
CASP7 P55210 1/20 0.56
NFKB2 Q00653 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7003777 0.84 ALDH1A1 (0.62) ALDH1A1HPGDKDM4ELMNARAB9A
SCHEMBL16246255 0.81 HPGD (0.59) ALDH1A1HPGDKDM4ELMNARAB9A
SCHEMBL7002469 0.80 ALDH1A1 (0.60) ALDH1A1HPGDKDM4ELMNARAB9A
SCHEMBL4140802 0.79 KMT2A (0.56) ALDH1A1HPGDKDM4ELMNARAB9A
SCHEMBL16263740 0.77 ALDH1A1 (0.54) ALDH1A1HPGDKDM4ELMNARAB9A
SCHEMBL31700539 0.77 ALDH1A1 (0.84) ALDH1A1HPGDKDM4ELMNARAB9A
SCHEMBL16246265 0.76 MAPT (0.56) ALDH1A1HPGDKDM4ELMNARAB9A
SCHEMBL7003934 0.76 ALDH1A1 (0.70) ALDH1A1HPGDKDM4ELMNARAB9A
SCHEMBL7673789 0.75 ALDH1A1 (0.62) ALDH1A1HPGDKDM4ELMNARAB9A
SCHEMBL6999632 0.75 RAB9A (0.62) ALDH1A1HPGDKDM4ELMNARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005033102-A2 THIOPHENE-BASED COMPOUNDS EXHIBITING ATP-UTILIZING ENZYME INHIBITORY ACTIVITY, AND COMPOSITIONS, AND USES THEREOF AMPHORA DISCOVERY CORPORATION (US) 2005-04-14 WO disclosed