SCHEMBL8299455

SCHEMBL8299455

O=C(C(=O)N1CCN(Cc2ccccc2)CC1)N1CCNCC1

nearest known ligand 0.67

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.67
ALDH1A1 P00352 6/20 0.63
LMNA P02545 4/20 0.63
KMT2A Q03164 3/20 0.63
SMN1; SMN2 Q16637 4/20 0.59
KDM4E B2RXH2 3/20 0.57
MEN1 O00255 2/20 0.56
TSHR P16473 2/20 0.56
FAAH O00519 1/20 0.56
MAPK1 P28482 1/20 0.56
L3MBTL1 Q9Y468 1/20 0.56
HPGD P15428 1/20 0.56
HTT P42858 1/20 0.56
PHGDH O43175 1/20 0.54
MGLL Q99685 1/20 0.54
MAPT P10636 1/20 0.54
CYP2C9 P11712 1/20 0.53
CYP2C19 P33261 1/20 0.53
HIF1A Q16665 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10825084 0.90 ALDH1A1 (0.70) SIGMAR1ALDH1A1LMNAKMT2ASMN1; SMN2
Bicarbonate SCHEMBL21981463 0.85 SIGMAR1 (0.85) SIGMAR1ALDH1A1LMNAKMT2ASMN1; SMN2
SCHEMBL7573306 0.83 SIGMAR1 (0.96) SIGMAR1ALDH1A1LMNAKMT2AMEN1
SCHEMBL8145866 0.83 SIGMAR1 (0.96) SIGMAR1ALDH1A1LMNAKMT2AMEN1
Acetic Acid SCHEMBL7452259 0.82 SIGMAR1 (0.79) SIGMAR1ALDH1A1LMNAKMT2ASMN1; SMN2
Urea SCHEMBL6942597 0.82 SIGMAR1 (0.79) SIGMAR1ALDH1A1LMNAKMT2ASMN1; SMN2
SCHEMBL9538814 0.81 SIGMAR1 (0.92) SIGMAR1ALDH1A1LMNAKMT2AMEN1
SCHEMBL13185789 0.81 SIGMAR1 (0.72) SIGMAR1ALDH1A1LMNAKMT2ASMN1; SMN2
SCHEMBL6138636 0.81 SIGMAR1 (1.00) SIGMAR1ALDH1A1LMNAKMT2AMEN1
SCHEMBL152631 0.81 SIGMAR1 (1.00) SIGMAR1ALDH1A1LMNAKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0927170-A1 PIPERAZINO DERIVATIVES AS NEUROKININ ANTAGONISTS SCHERING CORPORATION (US) 1999-07-07 EP disclosed
WO-1998008826-A1 PIPERAZINO DERIVATIVES AS NEUROKININ ANTAGONISTS SCHERING CORPORATION (US) 1998-03-05 WO disclosed