SCHEMBL8302370

SCHEMBL8302370

COC(=O)/C=C(\N[C@H](C(N)=O)c1ccccc1)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 7/20 0.48
CYP2C9 P11712 5/20 0.48
CYP2C19 P33261 5/20 0.48
CYP1A2 P05177 4/20 0.48
TSHR P16473 3/20 0.48
CYP2D6 P10635 3/20 0.48
SMN1; SMN2 Q16637 1/20 0.42
MTTP P55157 3/20 0.40
CNR2 P34972 2/20 0.39
PDPK1 O15530 1/20 0.39
NR4A1 P22736 1/20 0.39
NR4A2 P43354 1/20 0.39
NR4A3 Q92570 1/20 0.39
LDHA P00338 1/20 0.39
LDHB P07195 1/20 0.39
GAA P10253 2/20 0.38
MAPK1 P28482 2/20 0.38
LMNA P02545 1/20 0.38
POLB P06746 1/20 0.38
MAPT P10636 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8302401 0.88 GPR88 (0.40) CYP3A4CYP2C9CYP2C19CYP1A2TSHR
SCHEMBL8303022 0.86 ALDH1A1 (0.46) CYP3A4GAAPOLBMAPTHTT
SCHEMBL8307199 0.75 TSHR (0.43) CYP3A4CYP2C9TSHRSMN1; SMN2MAPK1
SCHEMBL8306394 0.75 TACR3 (0.40) CYP3A4CYP2C9CYP2C19CYP1A2TSHR
SCHEMBL8302507 0.70 CNR2 (0.44) CYP3A4CYP2C9CYP2C19CYP1A2TSHR
SCHEMBL13683341 0.69 ALDH1A1 (0.46) CYP3A4CYP2C9CYP2C19CYP1A2TSHR
SCHEMBL8305547 0.69 CNR2 (0.45) CYP3A4CYP2C9CYP2C19CYP1A2TSHR
SCHEMBL8047986 0.69 NR4A1 (0.68) SMN1; SMN2NR4A1NR4A2NR4A3MAPT
SCHEMBL18653054 0.68 CYP2D6 (0.51) CYP3A4CYP2C9CYP2C19TSHRCYP2D6
SCHEMBL12682989 0.68 CYP2D6 (0.51) CYP3A4CYP2C9CYP2C19TSHRCYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004085661-A2 PROCESS TO CHIRAL BETA-AMINO ACID DERIVATIVES MERCK & CO., INC (US) 2004-10-07 WO disclosed