SCHEMBL8303022

SCHEMBL8303022

COC(=O)/C=C(\N[C@H](C(N)=O)c1ccccc1)c1ccc(OC)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.46
CYP3A4 P08684 1/20 0.46
GAA P10253 1/20 0.45
ATM Q13315 1/20 0.44
EPHX1 P07099 1/20 0.43
CES2 O00748 1/20 0.43
CES1 P23141 1/20 0.43
MAPT P10636 4/20 0.43
KDM4E B2RXH2 2/20 0.43
KMT2A Q03164 3/20 0.42
MEN1 O00255 2/20 0.42
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
POLB P06746 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
PARP1 P09874 1/20 0.42
PARP10 Q53GL7 1/20 0.42
PARP2 Q9UGN5 1/20 0.42
PARP4 Q9UKK3 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8302401 0.92 GPR88 (0.40) ALDH1A1CYP3A4GAAATMMAPT
SCHEMBL8302370 0.86 CYP3A4 (0.48) ALDH1A1CYP3A4GAAMAPTPOLB
SCHEMBL8307199 0.79 TSHR (0.43) ALDH1A1CYP3A4ATMMAPTKDM4E
SCHEMBL8306394 0.78 TACR3 (0.40) ALDH1A1CYP3A4EPHX1CES2CES1
SCHEMBL8302507 0.73 CNR2 (0.44) ALDH1A1CYP3A4GAAATMEPHX1
SCHEMBL18653054 0.72 CYP2D6 (0.51) ALDH1A1CYP3A4ATMEPHX1MAPT
SCHEMBL6661082 0.72 RAB9A (0.66) ALDH1A1CYP3A4GAACES2CES1
SCHEMBL6661088 0.72 RAB9A (0.66) ALDH1A1CYP3A4GAACES2CES1
SCHEMBL7933746 0.72 RAB9A (0.66) ALDH1A1CYP3A4GAACES2CES1
SCHEMBL12682989 0.72 CYP2D6 (0.51) ALDH1A1CYP3A4ATMEPHX1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004085661-A2 PROCESS TO CHIRAL BETA-AMINO ACID DERIVATIVES MERCK & CO., INC (US) 2004-10-07 WO disclosed