SCHEMBL8302401

SCHEMBL8302401

COC(=O)/C=C(\N[C@H](C(N)=O)c1ccccc1)c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR88 Q9GZN0 1/20 0.40
TSHR P16473 3/20 0.40
CYP3A4 P08684 3/20 0.40
ALDH1A1 P00352 2/20 0.40
CYP1A2 P05177 2/20 0.40
KDM4E B2RXH2 1/20 0.39
MAPT P10636 1/20 0.39
S1PR3 Q99500 1/20 0.39
POLB P06746 1/20 0.39
KMT2A Q03164 2/20 0.38
GAA P10253 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
CYP2C9 P11712 2/20 0.38
MAPK1 P28482 2/20 0.38
CYP2C19 P33261 1/20 0.38
CNR1 P21554 1/20 0.38
TACR3 P29371 1/20 0.38
ATM Q13315 1/20 0.37
PDGFRA P16234 1/20 0.37
MAPKAPK2 P49137 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8303022 0.92 ALDH1A1 (0.46) CYP3A4ALDH1A1KDM4EMAPTPOLB
SCHEMBL8302370 0.88 CYP3A4 (0.48) TSHRCYP3A4ALDH1A1CYP1A2MAPT
SCHEMBL8306394 0.85 TACR3 (0.40) GPR88TSHRCYP3A4ALDH1A1CYP1A2
SCHEMBL8307199 0.83 TSHR (0.43) GPR88TSHRCYP3A4ALDH1A1KDM4E
SCHEMBL8302507 0.77 CNR2 (0.44) GPR88TSHRCYP3A4ALDH1A1CYP1A2
SCHEMBL18653054 0.76 CYP2D6 (0.51) GPR88TSHRCYP3A4ALDH1A1MAPT
SCHEMBL12682989 0.76 CYP2D6 (0.51) GPR88TSHRCYP3A4ALDH1A1MAPT
SCHEMBL8303024 0.76 LTB4R (0.48) TSHRALDH1A1CYP1A2KDM4EMAPT
SCHEMBL19658438 0.72 LMNA (0.46) GPR88CYP3A4POLBCYP2C9MAPK1
SCHEMBL12880512 0.72 LMNA (0.46) GPR88CYP3A4POLBCYP2C9MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004085661-A2 PROCESS TO CHIRAL BETA-AMINO ACID DERIVATIVES MERCK & CO., INC (US) 2004-10-07 WO disclosed